TFF3 vs Endomorphin-1

Head-to-head comparison of TFF3 (Trefoil Factor 3 (intestinal trefoil factor)) and Endomorphin-1 (Tyr-Pro-Trp-Phe-NH2) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyTFF3Endomorphin-1
CategoryGastrointestinalPain Management
Full NameTrefoil Factor 3 (intestinal trefoil factor)Tyr-Pro-Trp-Phe-NH2
Molecular Weight6370 Da610.71 Da
Half-Lifeunknown; likely short in circulationMinutes in plasma
Amino Acids594
Typical Doseresearch-only; model-dependent microgram to milligram ranges0.1-10 ug per animal
RouteOral/IntrarectalIntrathecal / subcutaneous
Purity≥98%≥98%
Studies Count70600
Research StatusPre-clinicalPre-clinical

TFF3 Benefits

  • epithelial-restitution
  • mucus-support
  • wound-healing
  • barrier-stability

Endomorphin-1 Benefits

  • mu-opioid selectivity
  • potent antinociception
  • endogenous peptide scaffold
  • useful for receptor-discovery studies

TFF3 Dosing

preclinical dosing varies widely by model|local or systemic administration|repeated dosing for inflammatory injury studies

Endomorphin-1 Dosing

Intrathecal 0.1-10 ug per animal|Subcutaneous 0.1-5 ug per animal|In vitro 0.1-100 nM

TFF3 Side Effects

  • limited human dosing data
  • protein stability issues
  • potential immunogenicity with exogenous use

Endomorphin-1 Side Effects

  • respiratory depression at high exposure
  • sedation
  • tolerance and dependence potential

Research Overview

TFF3

TFF3 is a well-established mucosal repair factor in the literature, especially in the context of intestinal injury and inflammation. Experimental studies support a role in accelerating restitution and protecting the epithelial surface in gut disease models.

Endomorphin-1

Endomorphin-1 is a key research peptide in studies of endogenous mu-opioid signaling and spinal analgesia. Like other peptide analgesics, its main translational hurdles are enzymatic instability, limited oral bioavailability, and delivery across barriers.

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Common Stacking Partners

TFF3 stacks with:

probioticsmesalaminezinc-carnosine

Endomorphin-1 stacks with:

gabapentinketamine
IBDmucosal-healingepithelial-restitutionmucusbarrier-protectionmu-opioidendogenous-peptideanalgesiapain-modulation