TFF3 vs DADLE

Head-to-head comparison of TFF3 (Trefoil Factor 3 (intestinal trefoil factor)) and DADLE ([D-Ala2, D-Leu5]-enkephalin) — benefits, dosing, side effects, research data, and where to buy.

Research Score

TFF3
4.1
PropertyTFF3DADLE
CategoryGastrointestinalPain Management
Full NameTrefoil Factor 3 (intestinal trefoil factor)[D-Ala2, D-Leu5]-enkephalin
Molecular Weight6370 Da569.67 Da
Half-Lifeunknown; likely short in circulation5-20 minutes in plasma
Amino Acids595
Typical Doseresearch-only; model-dependent microgram to milligram ranges0.01-2 ug per animal
RouteOral/IntrarectalIntrathecal / intracerebroventricular
Purity≥98%≥98%
Studies Count70450
Research StatusPre-clinicalPre-clinical

TFF3 Benefits

  • epithelial-restitution
  • mucus-support
  • wound-healing
  • barrier-stability

DADLE Benefits

  • delta-opioid agonism
  • enhanced peptide stability
  • spinal analgesia models
  • research on tolerance mechanisms

TFF3 Dosing

preclinical dosing varies widely by model|local or systemic administration|repeated dosing for inflammatory injury studies

DADLE Dosing

Intrathecal 0.01-2 ug per animal|Intracerebroventricular 0.01-1 ug per animal|In vitro 0.1-50 nM

TFF3 Side Effects

  • limited human dosing data
  • protein stability issues
  • potential immunogenicity with exogenous use

DADLE Side Effects

  • sedation
  • motor suppression at higher doses
  • opioid tolerance with repeated exposure

Research Overview

TFF3

TFF3 is a well-established mucosal repair factor in the literature, especially in the context of intestinal injury and inflammation. Experimental studies support a role in accelerating restitution and protecting the epithelial surface in gut disease models.

DADLE

DADLE has been studied for analgesic, neuroprotective, and receptor-selective opioid effects in animal and tissue models. It remains important as a mechanistic probe because it is more stable than endogenous enkephalins but still peptide-like in its delivery constraints.

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Common Stacking Partners

TFF3 stacks with:

probioticsmesalaminezinc-carnosine

DADLE stacks with:

morphineketamine
IBDmucosal-healingepithelial-restitutionmucusbarrier-protectionenkephalin-analogdelta-opioidanalgesiapeptide-therapeutic