Neurotensin vs Endomorphin-1

Head-to-head comparison of Neurotensin (Neurotensin) and Endomorphin-1 (Tyr-Pro-Trp-Phe-NH2) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyNeurotensinEndomorphin-1
CategoryPain ManagementPain Management
Full NameNeurotensinTyr-Pro-Trp-Phe-NH2
Molecular Weight1672.94610.71 Da
Half-LifeminutesMinutes in plasma
Amino Acids134
Typical DoseN/A|N/A0.1-10 ug per animal
RouteIntranasal/experimental injectionIntrathecal / subcutaneous
Purity≥98%≥98%
Studies Count81600
Research StatusPre-clinicalPre-clinical

Neurotensin Benefits

  • antinociceptive signaling
  • descending pain modulation
  • preclinical pain research

Endomorphin-1 Benefits

  • mu-opioid selectivity
  • potent antinociception
  • endogenous peptide scaffold
  • useful for receptor-discovery studies

Neurotensin Dosing

N/A|N/A

Endomorphin-1 Dosing

Intrathecal 0.1-10 ug per animal|Subcutaneous 0.1-5 ug per animal|In vitro 0.1-100 nM

Neurotensin Side Effects

  • hypotension
  • nausea
  • hypothermia

Endomorphin-1 Side Effects

  • respiratory depression at high exposure
  • sedation
  • tolerance and dependence potential

Research Overview

Neurotensin

Neurotensin has reproducible analgesic and neuromodulatory effects in preclinical studies, especially in inflammatory and neuropathic pain paradigms. It is not a standard clinical analgesic, but it is a real non-opioid peptide with pain-relevant biology.

Endomorphin-1

Endomorphin-1 is a key research peptide in studies of endogenous mu-opioid signaling and spinal analgesia. Like other peptide analgesics, its main translational hurdles are enzymatic instability, limited oral bioavailability, and delivery across barriers.

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Common Stacking Partners

Neurotensin stacks with:

NTS

Endomorphin-1 stacks with:

gabapentinketamine
non-opioidneuropeptideanalgesicmu-opioidendogenous-peptideanalgesiapain-modulation