Neurotensin vs Met-enkephalin

Head-to-head comparison of Neurotensin (Neurotensin) and Met-enkephalin (Tyr-Gly-Gly-Phe-Met) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyNeurotensinMet-enkephalin
CategoryPain ManagementPain Management
Full NameNeurotensinTyr-Gly-Gly-Phe-Met
Molecular Weight1672.94573.67 Da
Half-Lifeminutes1-5 minutes in plasma
Amino Acids135
Typical DoseN/A|N/A0.1-5 ug per animal
RouteIntranasal/experimental injectionIntrathecal / intracerebroventricular
Purity≥98%≥98%
Studies Count811200
Research StatusPre-clinicalPre-clinical

Neurotensin Benefits

  • antinociceptive signaling
  • descending pain modulation
  • preclinical pain research

Met-enkephalin Benefits

  • endogenous opioid signaling
  • analgesic reference ligand
  • spinal antinociception
  • neurochemical pain-pathway probe

Neurotensin Dosing

N/A|N/A

Met-enkephalin Dosing

Intrathecal 0.1-5 ug per animal|Intracerebroventricular 0.1-2 ug per animal|In vitro 1-100 nM

Neurotensin Side Effects

  • hypotension
  • nausea
  • hypothermia

Met-enkephalin Side Effects

  • sedation at higher exposure
  • constipation-like opioid effects
  • rapid enzymatic degradation

Research Overview

Neurotensin

Neurotensin has reproducible analgesic and neuromodulatory effects in preclinical studies, especially in inflammatory and neuropathic pain paradigms. It is not a standard clinical analgesic, but it is a real non-opioid peptide with pain-relevant biology.

Met-enkephalin

Met-enkephalin has been extensively used in receptor pharmacology and nociception studies to map mu and delta opioid biology. The main limitation in translational work is very short half-life from peptidase cleavage and poor systemic stability.

Ready to buy?

Find both peptides from our verified, lab-tested vendors with purity certificates and third-party testing.

Common Stacking Partners

Neurotensin stacks with:

NTS

Met-enkephalin stacks with:

gabapentinketamine
non-opioidneuropeptideanalgesicopioid-peptideenkephalinmu-opioidanalgesia