Met-enkephalin vs Somatostatin

Head-to-head comparison of Met-enkephalin (Tyr-Gly-Gly-Phe-Met) and Somatostatin (Somatostatin-14) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyMet-enkephalinSomatostatin
CategoryPain ManagementPain Management
Full NameTyr-Gly-Gly-Phe-MetSomatostatin-14
Molecular Weight573.67 Da1637.85
Half-Life1-5 minutes in plasma1-3 min
Amino Acids514
Typical Dose0.1-5 ug per animalN/A|N/A
RouteIntrathecal / intracerebroventricularIV/SC
Purity≥98%≥98%
Studies Count120084
Research StatusPre-clinicalApproved

Met-enkephalin Benefits

  • endogenous opioid signaling
  • analgesic reference ligand
  • spinal antinociception
  • neurochemical pain-pathway probe

Somatostatin Benefits

  • nociceptive inhibition
  • anti-inflammatory signaling
  • visceral pain modulation

Met-enkephalin Dosing

Intrathecal 0.1-5 ug per animal|Intracerebroventricular 0.1-2 ug per animal|In vitro 1-100 nM

Somatostatin Dosing

N/A|N/A

Met-enkephalin Side Effects

  • sedation at higher exposure
  • constipation-like opioid effects
  • rapid enzymatic degradation

Somatostatin Side Effects

  • hyperglycemia
  • bradycardia
  • GI upset

Research Overview

Met-enkephalin

Met-enkephalin has been extensively used in receptor pharmacology and nociception studies to map mu and delta opioid biology. The main limitation in translational work is very short half-life from peptidase cleavage and poor systemic stability.

Somatostatin

Somatostatin reduces release of multiple excitatory mediators and can suppress pain signaling in preclinical and limited translational work. Its analgesic use is not standard, but the peptide is real and mechanistically relevant to pain control.

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Common Stacking Partners

Met-enkephalin stacks with:

gabapentinketamine

Somatostatin stacks with:

SRIFGrowth hormone-inhibiting hormone
opioid-peptideenkephalinmu-opioidanalgesianon-opioidanalgesichormone