Metformin vs Melatonin

Head-to-head comparison of Metformin (Metformin Hydrochloride) and Melatonin (N-acetyl-5-methoxytryptamine) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyMetforminMelatonin
CategoryAnti-AgingAnti-Aging
Full NameMetformin HydrochlorideN-acetyl-5-methoxytryptamine
Molecular Weight165.63 Da232.28 Da
Half-Life4-8.7 hours20-50 minutes
Amino AcidsN/A0
Typical Dose500-2000 mg/day
RouteOral
Purity≥98%≥98%
Studies Count400015000
Research StatusClinicalApproved

Metformin Benefits

  • AMPK activation
  • improved insulin sensitivity
  • reduced oxidative stress
  • population-level longevity signal

Melatonin Benefits

  • Sleep regulation, circadian rhythm restoration, antioxidant protection, immune system support, potential neuroprotection, anti-aging effects

Metformin Dosing

500-2000 mg/day oral|start low and titrate in trials|taken with meals

Melatonin Dosing

0.5-10mg orally, typically 30-60 minutes before desired sleep time. Lower doses (0.5-3mg) often more effective for sleep onset

Metformin Side Effects

  • gastrointestinal upset
  • vitamin B12 reduction
  • diarrhea
  • rare lactic acidosis

Melatonin Side Effects

  • Drowsiness, headache, dizziness, nausea, vivid dreams, potential hormone interactions, daytime fatigue with higher doses

Research Overview

Metformin

Metformin has extensive human data and remains a leading candidate in geroscience research. Observational and mechanistic studies suggest it may influence pathways tied to aging, though definitive anti-longevity proof in healthy humans is still lacking.

Melatonin

Melatonin has extensive clinical research supporting its efficacy for sleep disorders, jet lag, and shift work sleep disorder. Emerging research investigates its potential anti-aging, neuroprotective, and immune-modulating properties with promising preliminary results.

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Common Stacking Partners

Metformin stacks with:

RapamycinNMNSpermidine

Melatonin stacks with:

MagnesiumL-TheanineGABAGlycine5-HTP
AMPKinsulin-sensitivitygerosciencemetabolismhormonesleepcircadianantioxidantneuroprotection