Larazotide vs TFF3

Head-to-head comparison of Larazotide (Larazotide acetate (AT-1001)) and TFF3 (Trefoil Factor 3 (intestinal trefoil factor)) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyLarazotideTFF3
CategoryGastrointestinalGastrointestinal
Full NameLarazotide acetate (AT-1001)Trefoil Factor 3 (intestinal trefoil factor)
Molecular WeightN/A6370 Da
Half-Lifeshort; designed for local gut actionunknown; likely short in circulation
Amino Acids859
Typical Dose0.5-4 mg TID (clinical studies)research-only; model-dependent microgram to milligram ranges
RouteOralOral/Intrarectal
Purity≥98%≥98%
Studies Count4070
Research StatusClinicalPre-clinical

Larazotide Benefits

  • tight-junction-support
  • reduced-permeability
  • symptom-reduction
  • barrier-protection

TFF3 Benefits

  • epithelial-restitution
  • mucus-support
  • wound-healing
  • barrier-stability

Larazotide Dosing

0.5-4 mg orally before meals in clinical trials|typically three times daily|short-course or chronic study protocols

TFF3 Dosing

preclinical dosing varies widely by model|local or systemic administration|repeated dosing for inflammatory injury studies

Larazotide Side Effects

  • headache
  • nausea
  • abdominal discomfort

TFF3 Side Effects

  • limited human dosing data
  • protein stability issues
  • potential immunogenicity with exogenous use

Research Overview

Larazotide

Clinical and translational studies suggest larazotide can reduce antigen passage across the epithelium and improve gut barrier function. It is one of the better-known peptides for intestinal permeability and barrier-focused gastrointestinal therapy.

TFF3

TFF3 is a well-established mucosal repair factor in the literature, especially in the context of intestinal injury and inflammation. Experimental studies support a role in accelerating restitution and protecting the epithelial surface in gut disease models.

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Common Stacking Partners

Larazotide stacks with:

gluten-free dietprobioticsmesalamine

TFF3 stacks with:

probioticsmesalaminezinc-carnosine
IBSceliactight-junctionspermeabilitybarrier-protectionIBDmucosal-healingepithelial-restitutionmucus