Huwentoxin-IV vs RgIA

Head-to-head comparison of Huwentoxin-IV (Huwentoxin-IV from Selenocosmia huwena venom) and RgIA (alpha-Conotoxin RgIA from Conus regius venom) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyHuwentoxin-IVRgIA
CategoryExperimentalExperimental
Full NameHuwentoxin-IV from Selenocosmia huwena venomalpha-Conotoxin RgIA from Conus regius venom
Molecular Weight4,000 Da1,670 Da
Half-LifeMinutes to hoursMinutes to hours
Amino Acids3513
Typical Dose0.01-1 nmol intrathecal|1-100 nM in vitro|single-dose rodent studies10-300 pmol intrathecal|1-100 nM in vitro|single-dose rodent studies
RouteIntrathecalIntrathecal
Purity≥98%≥98%
Studies Count110130
Research StatusPre-clinicalPre-clinical

Huwentoxin-IV Benefits

  • Nav1.7 selectivity
  • pain-channel validation
  • action-potential research
  • analgesic lead optimization

RgIA Benefits

  • alpha9alpha10 nAChR selectivity
  • neuropathic pain model tool
  • neuroimmune signaling research
  • analgesic lead discovery

Huwentoxin-IV Dosing

In vitro Nav1.7 electrophysiology|Intrathecal rodent analgesia studies|Single-bolus channel selectivity assays

RgIA Dosing

Intrathecal bolus in rodent pain models|Patch-clamp assays on alpha9alpha10 receptors|Single-dose pre-clinical screening

Huwentoxin-IV Side Effects

  • Neurological impairment at high exposure
  • off-target sodium-channel effects
  • injection-site irritation

RgIA Side Effects

  • Transient autonomic effects
  • off-target nicotinic blockade
  • injection-site irritation

Research Overview

Huwentoxin-IV

Studies show huwentoxin-IV can inhibit sodium-channel currents with notable selectivity, making it useful for dissecting pain-sensing neuron excitability. It is one of the better known spider-venom templates for Nav1.7-targeted drug discovery.

RgIA

Scientific studies show RgIA can strongly inhibit alpha9alpha10 nicotinic signaling with high selectivity compared with many other nAChR ligands. It is widely used to probe peripheral sensory pathways and inflammation-linked pain mechanisms.

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Common Stacking Partners

Huwentoxin-IV stacks with:

pregabalinlidocainemorphine

RgIA stacks with:

gabapentinpregabalinduloxetine
spider-venomsodium-channelnav1.7pain-researchcone-snailvenom-peptidenicotinic-receptor