Huwentoxin-IV vs Mambalgin-1

Head-to-head comparison of Huwentoxin-IV (Huwentoxin-IV from Selenocosmia huwena venom) and Mambalgin-1 (Mambalgin-1 from Dendroaspis polylepis venom) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyHuwentoxin-IVMambalgin-1
CategoryExperimentalExperimental
Full NameHuwentoxin-IV from Selenocosmia huwena venomMambalgin-1 from Dendroaspis polylepis venom
Molecular Weight4,000 Da6,300 Da
Half-LifeMinutes to hoursMinutes to hours
Amino Acids3557
Typical Dose0.01-1 nmol intrathecal|1-100 nM in vitro|single-dose rodent studies0.1-1 nmol intrathecal|10-100 nM in vitro|single-dose rodent studies
RouteIntrathecalIntrathecal
Purity≥98%≥98%
Studies Count11055
Research StatusPre-clinicalPre-clinical

Huwentoxin-IV Benefits

  • Nav1.7 selectivity
  • pain-channel validation
  • action-potential research
  • analgesic lead optimization

Mambalgin-1 Benefits

  • ASIC channel inhibition
  • non-opioid analgesia research
  • sensory-neuron physiology
  • lead optimization for pain therapeutics

Huwentoxin-IV Dosing

In vitro Nav1.7 electrophysiology|Intrathecal rodent analgesia studies|Single-bolus channel selectivity assays

Mambalgin-1 Dosing

Intrathecal pain-behavior studies|ASIC1a/ASIC1b electrophysiology|Acute dosing in rodents

Huwentoxin-IV Side Effects

  • Neurological impairment at high exposure
  • off-target sodium-channel effects
  • injection-site irritation

Mambalgin-1 Side Effects

  • Hypoactivity at high dose
  • off-target ASIC blockade
  • local irritation

Research Overview

Huwentoxin-IV

Studies show huwentoxin-IV can inhibit sodium-channel currents with notable selectivity, making it useful for dissecting pain-sensing neuron excitability. It is one of the better known spider-venom templates for Nav1.7-targeted drug discovery.

Mambalgin-1

Pre-clinical work shows mambalgin-1 can reduce pain behaviors by modulating proton-gated ion channels in peripheral and central pathways. It has become an important template for developing ASIC-targeted analgesics.

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Common Stacking Partners

Huwentoxin-IV stacks with:

pregabalinlidocainemorphine

Mambalgin-1 stacks with:

gabapentinbaclofenlidocaine
spider-venomsodium-channelnav1.7pain-researchsnake-venomthree-finger-toxinasic-blocker