Huwentoxin-IV vs Conantokin-G

Head-to-head comparison of Huwentoxin-IV (Huwentoxin-IV from Selenocosmia huwena venom) and Conantokin-G (Conantokin-G from Conus geographus venom) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyHuwentoxin-IVConantokin-G
CategoryExperimentalExperimental
Full NameHuwentoxin-IV from Selenocosmia huwena venomConantokin-G from Conus geographus venom
Molecular Weight4,000 Da2,150 Da
Half-LifeMinutes to hoursMinutes to hours
Amino Acids3517
Typical Dose0.01-1 nmol intrathecal|1-100 nM in vitro|single-dose rodent studies0.1-10 nmol intrathecal|10-1000 nM in vitro|single-dose rodent studies
RouteIntrathecalIntrathecal
Purity≥98%≥98%
Studies Count11095
Research StatusPre-clinicalPre-clinical

Huwentoxin-IV Benefits

  • Nav1.7 selectivity
  • pain-channel validation
  • action-potential research
  • analgesic lead optimization

Conantokin-G Benefits

  • NMDA receptor antagonism
  • seizure-model research
  • excitatory neurotransmission mapping
  • pain-mechanism studies

Huwentoxin-IV Dosing

In vitro Nav1.7 electrophysiology|Intrathecal rodent analgesia studies|Single-bolus channel selectivity assays

Conantokin-G Dosing

Intrathecal administration in seizure/pain models|NMDA receptor assays|In vitro excitation studies

Huwentoxin-IV Side Effects

  • Neurological impairment at high exposure
  • off-target sodium-channel effects
  • injection-site irritation

Conantokin-G Side Effects

  • Sedation or dizziness in animals
  • motor effects at high exposure
  • off-target NMDA modulation

Research Overview

Huwentoxin-IV

Studies show huwentoxin-IV can inhibit sodium-channel currents with notable selectivity, making it useful for dissecting pain-sensing neuron excitability. It is one of the better known spider-venom templates for Nav1.7-targeted drug discovery.

Conantokin-G

Research has shown conantokin-G can suppress NMDA-mediated responses in a sequence- and modification-dependent manner. It remains a classic marine peptide tool for probing glutamatergic signaling and analgesia-related pathways.

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Common Stacking Partners

Huwentoxin-IV stacks with:

pregabalinlidocainemorphine

Conantokin-G stacks with:

ketaminememantinelamotrigine
spider-venomsodium-channelnav1.7pain-researchcone-snailvenom-peptidenmda-antagonistneuroscience