Cholecystokinin-8 vs Met-enkephalin

Head-to-head comparison of Cholecystokinin-8 (Cholecystokinin (sulfated C-terminal octapeptide, CCK-8)) and Met-enkephalin (Tyr-Gly-Gly-Phe-Met) — benefits, dosing, side effects, research data, and where to buy.

PropertyCholecystokinin-8Met-enkephalin
CategoryEndocrine PeptidesPain Management
Full NameCholecystokinin (sulfated C-terminal octapeptide, CCK-8)Tyr-Gly-Gly-Phe-Met
Molecular Weight1143.2 Da573.67 Da
Half-Life1-2 min1-5 minutes in plasma
Amino AcidsDY(SO3H)MGWMDF-NH25
Typical Dosephysiologic low-picomolar-nanomolar range|research-dependent0.1-5 ug per animal
Routeendogenous secretion|research IV/SCIntrathecal / intracerebroventricular
Purity≥98%≥98%
Studies Count971200
Research StatusEndogenousPre-clinical

Cholecystokinin-8 Benefits

  • gallbladder contraction
  • pancreatic enzyme release
  • satiety signaling

Met-enkephalin Benefits

  • endogenous opioid signaling
  • analgesic reference ligand
  • spinal antinociception
  • neurochemical pain-pathway probe

Cholecystokinin-8 Dosing

physiologic secretion|research-dependent

Met-enkephalin Dosing

Intrathecal 0.1-5 ug per animal|Intracerebroventricular 0.1-2 ug per animal|In vitro 1-100 nM

Cholecystokinin-8 Side Effects

  • abdominal cramping
  • nausea
  • biliary contraction

Met-enkephalin Side Effects

  • sedation at higher exposure
  • constipation-like opioid effects
  • rapid enzymatic degradation

Research Overview

Cholecystokinin-8

CCK-8 is a canonical gut hormone fragment with extensive documentation in digestive physiology and appetite control. Sulfation of the tyrosine residue is important for high-affinity receptor activity.

Met-enkephalin

Met-enkephalin has been extensively used in receptor pharmacology and nociception studies to map mu and delta opioid biology. The main limitation in translational work is very short half-life from peptidase cleavage and poor systemic stability.

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Common Stacking Partners

Cholecystokinin-8 stacks with:

gallbladderpancreassatiety

Met-enkephalin stacks with:

gabapentinketamine
gut-hormonesatiety-peptideendocrine-peptideopioid-peptideenkephalinmu-opioidanalgesia