Met-enkephalin vs Neurotensin

Head-to-head comparison of Met-enkephalin (Tyr-Gly-Gly-Phe-Met) and Neurotensin (Neurotensin) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyMet-enkephalinNeurotensin
CategoryPain ManagementPain Management
Full NameTyr-Gly-Gly-Phe-MetNeurotensin
Molecular Weight573.67 Da1672.94
Half-Life1-5 minutes in plasmaminutes
Amino Acids513
Typical Dose0.1-5 ug per animalN/A|N/A
RouteIntrathecal / intracerebroventricularIntranasal/experimental injection
Purity≥98%≥98%
Studies Count120081
Research StatusPre-clinicalPre-clinical

Met-enkephalin Benefits

  • endogenous opioid signaling
  • analgesic reference ligand
  • spinal antinociception
  • neurochemical pain-pathway probe

Neurotensin Benefits

  • antinociceptive signaling
  • descending pain modulation
  • preclinical pain research

Met-enkephalin Dosing

Intrathecal 0.1-5 ug per animal|Intracerebroventricular 0.1-2 ug per animal|In vitro 1-100 nM

Neurotensin Dosing

N/A|N/A

Met-enkephalin Side Effects

  • sedation at higher exposure
  • constipation-like opioid effects
  • rapid enzymatic degradation

Neurotensin Side Effects

  • hypotension
  • nausea
  • hypothermia

Research Overview

Met-enkephalin

Met-enkephalin has been extensively used in receptor pharmacology and nociception studies to map mu and delta opioid biology. The main limitation in translational work is very short half-life from peptidase cleavage and poor systemic stability.

Neurotensin

Neurotensin has reproducible analgesic and neuromodulatory effects in preclinical studies, especially in inflammatory and neuropathic pain paradigms. It is not a standard clinical analgesic, but it is a real non-opioid peptide with pain-relevant biology.

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Common Stacking Partners

Met-enkephalin stacks with:

gabapentinketamine

Neurotensin stacks with:

NTS
opioid-peptideenkephalinmu-opioidanalgesianon-opioidneuropeptideanalgesic