RgIA vs Huwentoxin-IV

Head-to-head comparison of RgIA (alpha-Conotoxin RgIA from Conus regius venom) and Huwentoxin-IV (Huwentoxin-IV from Selenocosmia huwena venom) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyRgIAHuwentoxin-IV
CategoryExperimentalExperimental
Full Namealpha-Conotoxin RgIA from Conus regius venomHuwentoxin-IV from Selenocosmia huwena venom
Molecular Weight1,670 Da4,000 Da
Half-LifeMinutes to hoursMinutes to hours
Amino Acids1335
Typical Dose10-300 pmol intrathecal|1-100 nM in vitro|single-dose rodent studies0.01-1 nmol intrathecal|1-100 nM in vitro|single-dose rodent studies
RouteIntrathecalIntrathecal
Purity≥98%≥98%
Studies Count130110
Research StatusPre-clinicalPre-clinical

RgIA Benefits

  • alpha9alpha10 nAChR selectivity
  • neuropathic pain model tool
  • neuroimmune signaling research
  • analgesic lead discovery

Huwentoxin-IV Benefits

  • Nav1.7 selectivity
  • pain-channel validation
  • action-potential research
  • analgesic lead optimization

RgIA Dosing

Intrathecal bolus in rodent pain models|Patch-clamp assays on alpha9alpha10 receptors|Single-dose pre-clinical screening

Huwentoxin-IV Dosing

In vitro Nav1.7 electrophysiology|Intrathecal rodent analgesia studies|Single-bolus channel selectivity assays

RgIA Side Effects

  • Transient autonomic effects
  • off-target nicotinic blockade
  • injection-site irritation

Huwentoxin-IV Side Effects

  • Neurological impairment at high exposure
  • off-target sodium-channel effects
  • injection-site irritation

Research Overview

RgIA

Scientific studies show RgIA can strongly inhibit alpha9alpha10 nicotinic signaling with high selectivity compared with many other nAChR ligands. It is widely used to probe peripheral sensory pathways and inflammation-linked pain mechanisms.

Huwentoxin-IV

Studies show huwentoxin-IV can inhibit sodium-channel currents with notable selectivity, making it useful for dissecting pain-sensing neuron excitability. It is one of the better known spider-venom templates for Nav1.7-targeted drug discovery.

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Common Stacking Partners

RgIA stacks with:

gabapentinpregabalinduloxetine

Huwentoxin-IV stacks with:

pregabalinlidocainemorphine
cone-snailvenom-peptidenicotinic-receptorpain-researchspider-venomsodium-channelnav1.7