RgIA vs Conantokin-G

Head-to-head comparison of RgIA (alpha-Conotoxin RgIA from Conus regius venom) and Conantokin-G (Conantokin-G from Conus geographus venom) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyRgIAConantokin-G
CategoryExperimentalExperimental
Full Namealpha-Conotoxin RgIA from Conus regius venomConantokin-G from Conus geographus venom
Molecular Weight1,670 Da2,150 Da
Half-LifeMinutes to hoursMinutes to hours
Amino Acids1317
Typical Dose10-300 pmol intrathecal|1-100 nM in vitro|single-dose rodent studies0.1-10 nmol intrathecal|10-1000 nM in vitro|single-dose rodent studies
RouteIntrathecalIntrathecal
Purity≥98%≥98%
Studies Count13095
Research StatusPre-clinicalPre-clinical

RgIA Benefits

  • alpha9alpha10 nAChR selectivity
  • neuropathic pain model tool
  • neuroimmune signaling research
  • analgesic lead discovery

Conantokin-G Benefits

  • NMDA receptor antagonism
  • seizure-model research
  • excitatory neurotransmission mapping
  • pain-mechanism studies

RgIA Dosing

Intrathecal bolus in rodent pain models|Patch-clamp assays on alpha9alpha10 receptors|Single-dose pre-clinical screening

Conantokin-G Dosing

Intrathecal administration in seizure/pain models|NMDA receptor assays|In vitro excitation studies

RgIA Side Effects

  • Transient autonomic effects
  • off-target nicotinic blockade
  • injection-site irritation

Conantokin-G Side Effects

  • Sedation or dizziness in animals
  • motor effects at high exposure
  • off-target NMDA modulation

Research Overview

RgIA

Scientific studies show RgIA can strongly inhibit alpha9alpha10 nicotinic signaling with high selectivity compared with many other nAChR ligands. It is widely used to probe peripheral sensory pathways and inflammation-linked pain mechanisms.

Conantokin-G

Research has shown conantokin-G can suppress NMDA-mediated responses in a sequence- and modification-dependent manner. It remains a classic marine peptide tool for probing glutamatergic signaling and analgesia-related pathways.

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Common Stacking Partners

RgIA stacks with:

gabapentinpregabalinduloxetine

Conantokin-G stacks with:

ketaminememantinelamotrigine
cone-snailvenom-peptidenicotinic-receptorpain-researchnmda-antagonistneuroscience