Huwentoxin-IV vs Didemnin B

Head-to-head comparison of Huwentoxin-IV (Huwentoxin-IV from Selenocosmia huwena venom) and Didemnin B (Didemnin B) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyHuwentoxin-IVDidemnin B
CategoryExperimentalExperimental
Full NameHuwentoxin-IV from Selenocosmia huwena venomDidemnin B
Molecular Weight4,000 Da1112.4 Da
Half-LifeMinutes to hoursN/A
Amino Acids35N/A
Typical Dose0.01-1 nmol intrathecal|1-100 nM in vitro|single-dose rodent studies0.05-2 mg/m2 IV in early trials
RouteIntrathecalIntravenous
Purity≥98%≥98%
Studies Count110120
Research StatusPre-clinicalClinical

Huwentoxin-IV Benefits

  • Nav1.7 selectivity
  • pain-channel validation
  • action-potential research
  • analgesic lead optimization

Didemnin B Benefits

  • antineoplastic
  • antiviral
  • pro-apoptotic
  • immunomodulatory

Huwentoxin-IV Dosing

In vitro Nav1.7 electrophysiology|Intrathecal rodent analgesia studies|Single-bolus channel selectivity assays

Didemnin B Dosing

historic IV phase I/II oncology regimens|dose escalation in early trials|no approved dosing regimen

Huwentoxin-IV Side Effects

  • Neurological impairment at high exposure
  • off-target sodium-channel effects
  • injection-site irritation

Didemnin B Side Effects

  • nausea
  • vomiting
  • myelosuppression

Research Overview

Huwentoxin-IV

Studies show huwentoxin-IV can inhibit sodium-channel currents with notable selectivity, making it useful for dissecting pain-sensing neuron excitability. It is one of the better known spider-venom templates for Nav1.7-targeted drug discovery.

Didemnin B

Didemnin B showed strong cytotoxic and antiviral activity in early literature and became an important scaffold for later marine drug development. Its clinical progress was limited by toxicity, but it remains highly cited as a foundational marine depsipeptide.

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Common Stacking Partners

Huwentoxin-IV stacks with:

pregabalinlidocainemorphine

Didemnin B stacks with:

cisplatindoxorubicingemcitabine
spider-venomsodium-channelnav1.7pain-researchmarine-derivedtunicatedepsipeptideantitumor