CardiovascularPre-clinical

5A

Apolipoprotein A-I mimetic peptide 5A

37 Amino Acids · MW: ~4100 Da

Amino Acids

37

Molecular Weight

~4100 Da

Half-life

Hours to days depending on formulation

Research Score

4.1

Studies

41

Storage

Store lyophilized at -20°C, reconstituted at 2-8°C

What is 5A?

5A is a bihelical apoA-I mimetic peptide developed to improve cholesterol handling and HDL functionality. It has been studied for anti-inflammatory and anti-atherogenic effects in lipid metabolism models.

Key Benefits & Mechanisms

promotes cholesterol efflux

improves HDL function

reduces vascular inflammation

may stabilize plaques

Research Summary

5A has been investigated as a smaller, engineered HDL-mimetic that can modulate lipid handling without being a full apolipoprotein. Preclinical literature supports effects on reverse cholesterol transport and inflammation-related atherosclerosis endpoints.