TFF3 vs P11-4

Head-to-head comparison of TFF3 (Trefoil Factor 3 (intestinal trefoil factor)) and P11-4 (Self-assembling peptide P11-4 (Ac-QQRFEWEFEQQ-NH2)) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyTFF3P11-4
CategoryGastrointestinalDental & Oral
Full NameTrefoil Factor 3 (intestinal trefoil factor)Self-assembling peptide P11-4 (Ac-QQRFEWEFEQQ-NH2)
Molecular Weight6370 Da1466 Da
Half-Lifeunknown; likely short in circulationlocal activity for hours; peptide degraded over time
Amino Acids5911
Typical Doseresearch-only; model-dependent microgram to milligram ranges0.5-5 mg per lesion
RouteOral/IntrarectalTopical/Intraoral
Purity≥98%≥98%
Studies Count7040
Research StatusPre-clinicalClinical

TFF3 Benefits

  • epithelial-restitution
  • mucus-support
  • wound-healing
  • barrier-stability

P11-4 Benefits

  • enamel remineralization
  • early caries arrest
  • biomimetic scaffold formation
  • minimally invasive repair

TFF3 Dosing

preclinical dosing varies widely by model|local or systemic administration|repeated dosing for inflammatory injury studies

P11-4 Dosing

topical application to cleaned lesion|single-visit in-office application|repeat at follow-up if indicated

TFF3 Side Effects

  • limited human dosing data
  • protein stability issues
  • potential immunogenicity with exogenous use

P11-4 Side Effects

  • transient tooth sensitivity
  • local irritation
  • taste disturbance

Research Overview

TFF3

TFF3 is a well-established mucosal repair factor in the literature, especially in the context of intestinal injury and inflammation. Experimental studies support a role in accelerating restitution and protecting the epithelial surface in gut disease models.

P11-4

P11-4 has been studied for its ability to penetrate initial carious lesions and self-assemble into a fibrillar matrix that nucleates hydroxyapatite. Human and preclinical studies support its role in non-invasive enamel repair.

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Common Stacking Partners

TFF3 stacks with:

probioticsmesalaminezinc-carnosine

P11-4 stacks with:

fluoride varnishCPP-ACPxylitol
IBDmucosal-healingepithelial-restitutionmucusbarrier-protectionenamel-remineralizationcariesbiomimetic-peptideoral-health