Somatostatin vs Endomorphin-1

Head-to-head comparison of Somatostatin (Somatostatin-14) and Endomorphin-1 (Tyr-Pro-Trp-Phe-NH2) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertySomatostatinEndomorphin-1
CategoryPain ManagementPain Management
Full NameSomatostatin-14Tyr-Pro-Trp-Phe-NH2
Molecular Weight1637.85610.71 Da
Half-Life1-3 minMinutes in plasma
Amino Acids144
Typical DoseN/A|N/A0.1-10 ug per animal
RouteIV/SCIntrathecal / subcutaneous
Purity≥98%≥98%
Studies Count84600
Research StatusApprovedPre-clinical

Somatostatin Benefits

  • nociceptive inhibition
  • anti-inflammatory signaling
  • visceral pain modulation

Endomorphin-1 Benefits

  • mu-opioid selectivity
  • potent antinociception
  • endogenous peptide scaffold
  • useful for receptor-discovery studies

Somatostatin Dosing

N/A|N/A

Endomorphin-1 Dosing

Intrathecal 0.1-10 ug per animal|Subcutaneous 0.1-5 ug per animal|In vitro 0.1-100 nM

Somatostatin Side Effects

  • hyperglycemia
  • bradycardia
  • GI upset

Endomorphin-1 Side Effects

  • respiratory depression at high exposure
  • sedation
  • tolerance and dependence potential

Research Overview

Somatostatin

Somatostatin reduces release of multiple excitatory mediators and can suppress pain signaling in preclinical and limited translational work. Its analgesic use is not standard, but the peptide is real and mechanistically relevant to pain control.

Endomorphin-1

Endomorphin-1 is a key research peptide in studies of endogenous mu-opioid signaling and spinal analgesia. Like other peptide analgesics, its main translational hurdles are enzymatic instability, limited oral bioavailability, and delivery across barriers.

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Common Stacking Partners

Somatostatin stacks with:

SRIFGrowth hormone-inhibiting hormone

Endomorphin-1 stacks with:

gabapentinketamine
non-opioidanalgesichormonemu-opioidendogenous-peptideanalgesiapain-modulation