Roxadustat vs FS315

Head-to-head comparison of Roxadustat (Roxadustat (FG-4592), hypoxia-inducible factor prolyl hydroxylase inhibitor) and FS315 (Follistatin-315 (FS315)) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyRoxadustatFS315
CategoryMuscle & PerformanceMuscle & Performance
Full NameRoxadustat (FG-4592), hypoxia-inducible factor prolyl hydroxylase inhibitorFollistatin-315 (FS315)
Molecular Weight352.35 Da~40 kDa
Half-Life~12-16 hN/A; depends on construct/delivery
Amino AcidsN/A315
Typical Dose70-100 mg orally three times weeklyResearch-only; no standardized human dose
RouteOralIntramuscular / research expression systems
Purity≥98%≥98%
Studies Count18095
Research StatusClinicalPre-clinical

Roxadustat Benefits

  • induces endogenous EPO
  • improves iron handling
  • raises hemoglobin
  • may improve exercise tolerance

FS315 Benefits

  • activin neutralization
  • muscle growth signaling
  • anti-catabolic support
  • tissue repair modulation

Roxadustat Dosing

70-100 mg orally 3x weekly|Titrate by hemoglobin response|Monitor iron indices regularly

FS315 Dosing

Research-only recombinant/protein-expression studies|no standardized clinical dose|route varies by platform

Roxadustat Side Effects

  • nausea
  • hypertension
  • thrombotic events

FS315 Side Effects

  • off-target endocrine effects
  • immune response risk
  • fluid balance changes

Research Overview

Roxadustat

Large clinical studies support roxadustat for anemia, especially in chronic kidney disease populations. Direct VO2 max enhancement data in healthy athletes are limited, so its performance effects remain mostly inferential.

FS315

Follistatin-315 is a key reference isoform in studies of muscle anabolism and reproductive/endocrine biology. In muscle research, it is relevant because it suppresses activin and can indirectly blunt myostatin pathway output.

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Common Stacking Partners

Roxadustat stacks with:

IronFolate

FS315 stacks with:

CreatineVitamin DLeucine
hif-stabilizererythropoiesisvo2-maxoralfollistatinactivin-inhibitormyostatin-pathwayprotein