Melatonin vs Metformin

Head-to-head comparison of Melatonin (N-acetyl-5-methoxytryptamine) and Metformin (Metformin Hydrochloride) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyMelatoninMetformin
CategoryAnti-AgingAnti-Aging
Full NameN-acetyl-5-methoxytryptamineMetformin Hydrochloride
Molecular Weight232.28 Da165.63 Da
Half-Life20-50 minutes4-8.7 hours
Amino Acids0N/A
Typical Dose500-2000 mg/day
RouteOral
Purity≥98%≥98%
Studies Count150004000
Research StatusApprovedClinical

Melatonin Benefits

  • Sleep regulation, circadian rhythm restoration, antioxidant protection, immune system support, potential neuroprotection, anti-aging effects

Metformin Benefits

  • AMPK activation
  • improved insulin sensitivity
  • reduced oxidative stress
  • population-level longevity signal

Melatonin Dosing

0.5-10mg orally, typically 30-60 minutes before desired sleep time. Lower doses (0.5-3mg) often more effective for sleep onset

Metformin Dosing

500-2000 mg/day oral|start low and titrate in trials|taken with meals

Melatonin Side Effects

  • Drowsiness, headache, dizziness, nausea, vivid dreams, potential hormone interactions, daytime fatigue with higher doses

Metformin Side Effects

  • gastrointestinal upset
  • vitamin B12 reduction
  • diarrhea
  • rare lactic acidosis

Research Overview

Melatonin

Melatonin has extensive clinical research supporting its efficacy for sleep disorders, jet lag, and shift work sleep disorder. Emerging research investigates its potential anti-aging, neuroprotective, and immune-modulating properties with promising preliminary results.

Metformin

Metformin has extensive human data and remains a leading candidate in geroscience research. Observational and mechanistic studies suggest it may influence pathways tied to aging, though definitive anti-longevity proof in healthy humans is still lacking.

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Common Stacking Partners

Melatonin stacks with:

MagnesiumL-TheanineGABAGlycine5-HTP

Metformin stacks with:

RapamycinNMNSpermidine
hormonesleepcircadianantioxidantneuroprotectionAMPKinsulin-sensitivitygerosciencemetabolism