Metformin vs Fisetin

Head-to-head comparison of Metformin (Metformin Hydrochloride) and Fisetin (3,3',4',7-Tetrahydroxyflavone) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyMetforminFisetin
CategoryAnti-AgingAnti-Aging
Full NameMetformin Hydrochloride3,3',4',7-Tetrahydroxyflavone
Molecular Weight165.63 Da286.24 Da
Half-Life4-8.7 hours3-8 hours
Amino AcidsN/AN/A
Typical Dose500-2000 mg/day1000-2000 mg/day
RouteOralOral
Purity≥98%≥98%
Studies Count4000180
Research StatusClinicalPre-clinical

Metformin Benefits

  • AMPK activation
  • improved insulin sensitivity
  • reduced oxidative stress
  • population-level longevity signal

Fisetin Benefits

  • senolytic activity
  • reduces inflammatory signaling
  • supports mitochondrial function
  • may improve healthspan

Metformin Dosing

500-2000 mg/day oral|start low and titrate in trials|taken with meals

Fisetin Dosing

1000-2000 mg/day orally|1-2 days per month in senolytic-style studies|take with a fat-containing meal

Metformin Side Effects

  • gastrointestinal upset
  • vitamin B12 reduction
  • diarrhea
  • rare lactic acidosis

Fisetin Side Effects

  • GI upset
  • headache
  • possible blood-thinner interaction

Research Overview

Metformin

Metformin has extensive human data and remains a leading candidate in geroscience research. Observational and mechanistic studies suggest it may influence pathways tied to aging, though definitive anti-longevity proof in healthy humans is still lacking.

Fisetin

Preclinical studies show fisetin can selectively target senescent cells and reduce age-related inflammatory markers. Early human research exists, but definitive anti-aging outcomes in humans are still unproven.

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Common Stacking Partners

Metformin stacks with:

RapamycinNMNSpermidine

Fisetin stacks with:

QuercetinCoQ10Nicotinamide Riboside
AMPKinsulin-sensitivitygerosciencemetabolismsenolyticpolyphenolantioxidanthealthspan