Larazotide vs Histatin-5

Head-to-head comparison of Larazotide (Larazotide acetate (AT-1001)) and Histatin-5 (Human histatin 5) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyLarazotideHistatin-5
CategoryGastrointestinalDental & Oral
Full NameLarazotide acetate (AT-1001)Human histatin 5
Molecular WeightN/A3035 Da
Half-Lifeshort; designed for local gut actionminutes in saliva
Amino Acids824
Typical Dose0.5-4 mg TID (clinical studies)1-100 µM in research formulations
RouteOralTopical/Oral rinse
Purity≥98%≥98%
Studies Count40120
Research StatusClinicalPre-clinical

Larazotide Benefits

  • tight-junction-support
  • reduced-permeability
  • symptom-reduction
  • barrier-protection

Histatin-5 Benefits

  • anti-Candida activity
  • biofilm suppression
  • mucosal wound support
  • oral innate immunity

Larazotide Dosing

0.5-4 mg orally before meals in clinical trials|typically three times daily|short-course or chronic study protocols

Histatin-5 Dosing

topical rinse or gel|short contact exposure|repeat applications in research protocols

Larazotide Side Effects

  • headache
  • nausea
  • abdominal discomfort

Histatin-5 Side Effects

  • local irritation
  • proteolytic instability
  • dose-dependent cytotoxicity in vitro

Research Overview

Larazotide

Clinical and translational studies suggest larazotide can reduce antigen passage across the epithelium and improve gut barrier function. It is one of the better-known peptides for intestinal permeability and barrier-focused gastrointestinal therapy.

Histatin-5

Histatin-5 is a major salivary defense peptide that can kill Candida species and influence oral microbial communities. It is also investigated for wound-healing and xerostomia-associated oral infection models.

Ready to buy?

Find both peptides from our verified, lab-tested vendors with purity certificates and third-party testing.

Common Stacking Partners

Larazotide stacks with:

gluten-free dietprobioticsmesalamine

Histatin-5 stacks with:

chlorhexidinefluoridexylitol
IBSceliactight-junctionspermeabilitybarrier-protectionantimicrobial-peptidecandidasalivaoral-defense