Didemnin B vs Huwentoxin-IV

Head-to-head comparison of Didemnin B (Didemnin B) and Huwentoxin-IV (Huwentoxin-IV from Selenocosmia huwena venom) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyDidemnin BHuwentoxin-IV
CategoryExperimentalExperimental
Full NameDidemnin BHuwentoxin-IV from Selenocosmia huwena venom
Molecular Weight1112.4 Da4,000 Da
Half-LifeN/AMinutes to hours
Amino AcidsN/A35
Typical Dose0.05-2 mg/m2 IV in early trials0.01-1 nmol intrathecal|1-100 nM in vitro|single-dose rodent studies
RouteIntravenousIntrathecal
Purity≥98%≥98%
Studies Count120110
Research StatusClinicalPre-clinical

Didemnin B Benefits

  • antineoplastic
  • antiviral
  • pro-apoptotic
  • immunomodulatory

Huwentoxin-IV Benefits

  • Nav1.7 selectivity
  • pain-channel validation
  • action-potential research
  • analgesic lead optimization

Didemnin B Dosing

historic IV phase I/II oncology regimens|dose escalation in early trials|no approved dosing regimen

Huwentoxin-IV Dosing

In vitro Nav1.7 electrophysiology|Intrathecal rodent analgesia studies|Single-bolus channel selectivity assays

Didemnin B Side Effects

  • nausea
  • vomiting
  • myelosuppression

Huwentoxin-IV Side Effects

  • Neurological impairment at high exposure
  • off-target sodium-channel effects
  • injection-site irritation

Research Overview

Didemnin B

Didemnin B showed strong cytotoxic and antiviral activity in early literature and became an important scaffold for later marine drug development. Its clinical progress was limited by toxicity, but it remains highly cited as a foundational marine depsipeptide.

Huwentoxin-IV

Studies show huwentoxin-IV can inhibit sodium-channel currents with notable selectivity, making it useful for dissecting pain-sensing neuron excitability. It is one of the better known spider-venom templates for Nav1.7-targeted drug discovery.

Ready to buy?

Find both peptides from our verified, lab-tested vendors with purity certificates and third-party testing.

Common Stacking Partners

Didemnin B stacks with:

cisplatindoxorubicingemcitabine

Huwentoxin-IV stacks with:

pregabalinlidocainemorphine
marine-derivedtunicatedepsipeptideantitumorspider-venomsodium-channelnav1.7pain-research