DADLE vs Insulin Glargine

Head-to-head comparison of DADLE ([D-Ala2, D-Leu5]-enkephalin) and Insulin Glargine (Insulin glargine (A21Gly,B31Arg,B32Arg human insulin analog)) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyDADLEInsulin Glargine
CategoryPain ManagementDiabetes & Metabolic
Full Name[D-Ala2, D-Leu5]-enkephalinInsulin glargine (A21Gly,B31Arg,B32Arg human insulin analog)
Molecular Weight569.67 Da6063.6 Da
Half-Life5-20 minutes in plasmaAbout 12-24 hours
Amino Acids551
Typical Dose0.01-2 ug per animal0.1-0.2 U/kg once daily
RouteIntrathecal / intracerebroventricularSubcutaneous
Purity≥98%≥98%
Studies Count45013000
Research StatusPre-clinicalApproved

DADLE Benefits

  • delta-opioid agonism
  • enhanced peptide stability
  • spinal analgesia models
  • research on tolerance mechanisms

Insulin Glargine Benefits

  • Once-daily basal coverage
  • Smooth action profile
  • Lower nocturnal hypoglycemia risk
  • Improves fasting glucose control

DADLE Dosing

Intrathecal 0.01-2 ug per animal|Intracerebroventricular 0.01-1 ug per animal|In vitro 0.1-50 nM

Insulin Glargine Dosing

Inject SC once daily at the same time each day|Titrate every 3-4 days to fasting glucose targets|Can be combined with prandial insulin

DADLE Side Effects

  • sedation
  • motor suppression at higher doses
  • opioid tolerance with repeated exposure

Insulin Glargine Side Effects

  • Hypoglycemia
  • Injection-site reactions
  • Weight gain

Research Overview

DADLE

DADLE has been studied for analgesic, neuroprotective, and receptor-selective opioid effects in animal and tissue models. It remains important as a mechanistic probe because it is more stable than endogenous enkephalins but still peptide-like in its delivery constraints.

Insulin Glargine

Clinical and translational studies support its use as a basal comparator because of prolonged absorption and stable glycemic control. It is heavily used in basal-bolus regimen research and insulin-delivery optimization studies.

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Common Stacking Partners

DADLE stacks with:

morphineketamine

Insulin Glargine stacks with:

Insulin LisproInsulin Aspart
enkephalin-analogdelta-opioidanalgesiapeptide-therapeuticbasal insulinlong-actingfasting glucose