Conantokin-G vs RgIA

Head-to-head comparison of Conantokin-G (Conantokin-G from Conus geographus venom) and RgIA (alpha-Conotoxin RgIA from Conus regius venom) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyConantokin-GRgIA
CategoryExperimentalExperimental
Full NameConantokin-G from Conus geographus venomalpha-Conotoxin RgIA from Conus regius venom
Molecular Weight2,150 Da1,670 Da
Half-LifeMinutes to hoursMinutes to hours
Amino Acids1713
Typical Dose0.1-10 nmol intrathecal|10-1000 nM in vitro|single-dose rodent studies10-300 pmol intrathecal|1-100 nM in vitro|single-dose rodent studies
RouteIntrathecalIntrathecal
Purity≥98%≥98%
Studies Count95130
Research StatusPre-clinicalPre-clinical

Conantokin-G Benefits

  • NMDA receptor antagonism
  • seizure-model research
  • excitatory neurotransmission mapping
  • pain-mechanism studies

RgIA Benefits

  • alpha9alpha10 nAChR selectivity
  • neuropathic pain model tool
  • neuroimmune signaling research
  • analgesic lead discovery

Conantokin-G Dosing

Intrathecal administration in seizure/pain models|NMDA receptor assays|In vitro excitation studies

RgIA Dosing

Intrathecal bolus in rodent pain models|Patch-clamp assays on alpha9alpha10 receptors|Single-dose pre-clinical screening

Conantokin-G Side Effects

  • Sedation or dizziness in animals
  • motor effects at high exposure
  • off-target NMDA modulation

RgIA Side Effects

  • Transient autonomic effects
  • off-target nicotinic blockade
  • injection-site irritation

Research Overview

Conantokin-G

Research has shown conantokin-G can suppress NMDA-mediated responses in a sequence- and modification-dependent manner. It remains a classic marine peptide tool for probing glutamatergic signaling and analgesia-related pathways.

RgIA

Scientific studies show RgIA can strongly inhibit alpha9alpha10 nicotinic signaling with high selectivity compared with many other nAChR ligands. It is widely used to probe peripheral sensory pathways and inflammation-linked pain mechanisms.

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Common Stacking Partners

Conantokin-G stacks with:

ketaminememantinelamotrigine

RgIA stacks with:

gabapentinpregabalinduloxetine
cone-snailvenom-peptidenmda-antagonistneurosciencenicotinic-receptorpain-research