Cholecystokinin-8 vs Linaclotide

Head-to-head comparison of Cholecystokinin-8 (Cholecystokinin (sulfated C-terminal octapeptide, CCK-8)) and Linaclotide (Linaclotide) — benefits, dosing, side effects, research data, and where to buy.

PropertyCholecystokinin-8Linaclotide
CategoryEndocrine PeptidesGastrointestinal
Full NameCholecystokinin (sulfated C-terminal octapeptide, CCK-8)Linaclotide
Molecular Weight1143.2 Da1526.8 Da
Half-Life1-2 minActive locally; negligible systemic half-life
Amino AcidsDY(SO3H)MGWMDF-NH214
Typical Dosephysiologic low-picomolar-nanomolar range|research-dependent72-290 mcg once daily
Routeendogenous secretion|research IV/SCOral
Purity≥98%≥98%
Studies Count971200
Research StatusEndogenousClinical

Cholecystokinin-8 Benefits

  • gallbladder contraction
  • pancreatic enzyme release
  • satiety signaling

Linaclotide Benefits

  • improves-bowel-movements
  • reduces-abdominal-pain
  • increases-intestinal-secretion
  • supports-transit

Cholecystokinin-8 Dosing

physiologic secretion|research-dependent

Linaclotide Dosing

72 mcg PO daily|145 mcg PO daily|290 mcg PO daily

Cholecystokinin-8 Side Effects

  • abdominal cramping
  • nausea
  • biliary contraction

Linaclotide Side Effects

  • diarrhea
  • abdominal-pain
  • bloating

Research Overview

Cholecystokinin-8

CCK-8 is a canonical gut hormone fragment with extensive documentation in digestive physiology and appetite control. Sulfation of the tyrosine residue is important for high-affinity receptor activity.

Linaclotide

Linaclotide has extensive clinical evidence for chronic idiopathic constipation and IBS-C, with consistent effects on stool frequency and abdominal symptom relief. Its mechanism is local GC-C activation in the gut with minimal systemic exposure.

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Common Stacking Partners

Cholecystokinin-8 stacks with:

gallbladderpancreassatiety

Linaclotide stacks with:

dietary-fiberhydrationmagnesium
gut-hormonesatiety-peptideendocrine-peptideibs-cconstipationgc-c-agonistintestinal-secretion