Apratoxin A vs SNX-482

Head-to-head comparison of Apratoxin A (Apratoxin A) and SNX-482 (SNX-482 peptide from Hysterocrates gigas venom) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyApratoxin ASNX-482
CategoryExperimentalExperimental
Full NameApratoxin ASNX-482 peptide from Hysterocrates gigas venom
Molecular WeightN/A4,300 Da
Half-LifeN/AMinutes to hours
Amino AcidsN/A41
Typical DoseN/A in humans; nanomolar in vitro0.01-1 nmol intrathecal|1-100 nM in vitro|single-dose electrophysiology studies
RouteIntraperitoneal / Intravenous (preclinical)Intrathecal
Purity≥98%≥98%
Studies Count14085
Research StatusPre-clinicalPre-clinical

Apratoxin A Benefits

  • antineoplastic
  • anti-angiogenic
  • Sec61 inhibition
  • anti-proliferative

SNX-482 Benefits

  • Cav2.3 blockade
  • synaptic transmission studies
  • excitability mapping
  • pain and epilepsy research

Apratoxin A Dosing

preclinical in vitro nanomolar use|animal studies only|no human dosing established

SNX-482 Dosing

Patch-clamp Cav2.3 assays|Intrathecal neurophysiology studies|Acute channel-blockade experiments

Apratoxin A Side Effects

  • hepatotoxicity
  • general cytotoxicity
  • GI toxicity

SNX-482 Side Effects

  • Ataxia at high exposure
  • off-target calcium-channel block
  • cardiovascular effects in animal models

Research Overview

Apratoxin A

Apratoxin A is a well-studied lead compound for targeting secretory and membrane protein biogenesis in cancer cells. Medicinal chemistry programs around apratoxins focus on improving selectivity and reducing hepatotoxicity while preserving potency.

SNX-482

SNX-482 has been used to dissect R-type calcium currents in neurons and endocrine cells, and to map the role of Cav2.3 in excitability. Its selectivity profile has made it a standard research reagent in channel pharmacology.

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Common Stacking Partners

Apratoxin A stacks with:

gemcitabinedocetaxelEGFR inhibitors

SNX-482 stacks with:

gabapentinbaclofenketamine
marine-derivedcyanobacteriadepsipeptideSec61spider-venomcalcium-channelcav2.3neurophysiology