Drug DeliveryPre-clinical

TAT

HIV-1 TAT protein transduction domain

YGRKKRRQRRR Amino Acids · MW: 1560.9

Amino Acids

YGRKKRRQRRR

Molecular Weight

1560.9

Half-life

minutes to <1 h in serum; formulation-dependent

Research Score

4.6

Studies

92

Storage

Store lyophilized at -20°C, reconstituted at 2-8°C

What is TAT?

A classic cationic cell-penetrating peptide derived from the HIV-1 transactivator of transcription protein. It is widely used to ferry proteins, peptides, and nucleic acids into cells in preclinical drug-delivery studies.

Key Benefits & Mechanisms

high membrane translocation

broad cargo compatibility

well-characterized uptake biology

Research Summary

Extensively used as a modular CPP for intracellular delivery of proteins, siRNA, and nanoparticles; activity is often improved by cargo conjugation strategies and endosomal escape motifs.