Tesofensine vs Oxyntomodulin

Head-to-head comparison of Tesofensine (Tesofensine (NS2330)) and Oxyntomodulin (Endogenous glucagon-like peptide 1 and glucagon co-agonist peptide) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyTesofensineOxyntomodulin
CategoryWeight ManagementWeight Management
Full NameTesofensine (NS2330)Endogenous glucagon-like peptide 1 and glucagon co-agonist peptide
Molecular Weight426.52 g/mol~4,200 Da
Half-Life~200-300 hours12-15 minutes
Amino AcidsSmall molecule37
Typical DoseResearch doses vary; commonly 100-300 mcg in small human studies
RouteSubcutaneous/IV
Purity>98%≥98%
Studies Count3580
Research StatusPhase III Clinical TrialsClinical

Tesofensine Benefits

  • Potent appetite suppression, increased metabolic rate, enhanced thermogenesis, improved mood during dieting, reduces food reward-seeking behavior

Oxyntomodulin Benefits

  • reduces appetite
  • increases satiety
  • supports weight loss
  • improves postprandial metabolic signaling

Tesofensine Dosing

Clinical doses: 0.25-1.0 mg orally once daily. Research typically uses 0.5 mg. Extremely long half-life (8-13 days) means steady-state in 7-10 days.

Oxyntomodulin Dosing

Research-only dosing|Subcutaneous or IV administration in trials|Pair with calorie restriction and monitoring

Tesofensine Side Effects

  • Dry mouth, insomnia, constipation, increased heart rate, elevated blood pressure. Not recommended with uncontrolled hypertension.

Oxyntomodulin Side Effects

  • nausea
  • GI discomfort
  • decreased appetite beyond target

Research Overview

Tesofensine

Phase II trials showed 12.8 kg average weight loss at 1.0 mg dose over 6 months. Simultaneously inhibits reuptake of norepinephrine, dopamine, and serotonin, producing appetite suppression and increased thermogenesis.

Oxyntomodulin

Human studies showed acute reductions in food intake and modest weight loss, helping establish the GLP-1 and glucagon co-agonism concept. It remains a foundational peptide for obesity and satiety research.

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Common Stacking Partners

Tesofensine stacks with:

5-Amino-1MQAOD-9604MOTS-c

Oxyntomodulin stacks with:

calorie-deficitresistance-training
weight-lossappetite-suppressanttriple-reuptake-inhibitorthermogenesisGLP-1glucagon-coagonistendogenous-peptideappetite-regulation