Tesofensine vs Elamipretide

Head-to-head comparison of Tesofensine (Tesofensine (NS2330)) and Elamipretide (Elamipretide (MTP-131, SS-31)) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyTesofensineElamipretide
CategoryWeight ManagementMuscle & Performance
Full NameTesofensine (NS2330)Elamipretide (MTP-131, SS-31)
Molecular Weight426.52 g/mol639.8 Da
Half-Life~200-300 hours1-4 hours
Amino AcidsSmall molecule4
Typical Dose0.01-0.25 mg/kg/day
RouteSubcutaneous/Intravenous
Purity>98%≥98%
Studies Count35120
Research StatusPhase III Clinical TrialsClinical

Tesofensine Benefits

  • Potent appetite suppression, increased metabolic rate, enhanced thermogenesis, improved mood during dieting, reduces food reward-seeking behavior

Elamipretide Benefits

  • mitochondrial protection
  • reduced oxidative stress
  • improved fatigue resistance
  • may support exercise tolerance

Tesofensine Dosing

Clinical doses: 0.25-1.0 mg orally once daily. Research typically uses 0.5 mg. Extremely long half-life (8-13 days) means steady-state in 7-10 days.

Elamipretide Dosing

0.01-0.25 mg/kg/day SC (clinical research)|daily dosing in trials|alternative IV protocols in some studies

Tesofensine Side Effects

  • Dry mouth, insomnia, constipation, increased heart rate, elevated blood pressure. Not recommended with uncontrolled hypertension.

Elamipretide Side Effects

  • nausea
  • injection-site reactions
  • diarrhea
  • headache

Research Overview

Tesofensine

Phase II trials showed 12.8 kg average weight loss at 1.0 mg dose over 6 months. Simultaneously inhibits reuptake of norepinephrine, dopamine, and serotonin, producing appetite suppression and increased thermogenesis.

Elamipretide

Clinical and translational studies show elamipretide can improve mitochondrial function and some functional endpoints in mitochondrial disorders. Skeletal muscle research suggests benefits are driven by energy metabolism rather than direct muscle-building effects.

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Common Stacking Partners

Tesofensine stacks with:

5-Amino-1MQAOD-9604MOTS-c

Elamipretide stacks with:

creatinecoenzyme-q10protein
weight-lossappetite-suppressanttriple-reuptake-inhibitorthermogenesismitochondriafatigueenergy-metabolismperformance