Tesofensine vs Arenicin-1

Head-to-head comparison of Tesofensine (Tesofensine (NS2330)) and Arenicin-1 (Arenicin-1) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyTesofensineArenicin-1
CategoryWeight ManagementMarine-Derived
Full NameTesofensine (NS2330)Arenicin-1
Molecular Weight426.52 g/mol2079 Da
Half-Life~200-300 hoursn/a
Amino AcidsSmall molecule21
Typical Dosen/a
Routepreclinical
Purity>98%≥98%
Studies Count3576
Research StatusPhase III Clinical TrialsPre-clinical

Tesofensine Benefits

  • Potent appetite suppression, increased metabolic rate, enhanced thermogenesis, improved mood during dieting, reduces food reward-seeking behavior

Arenicin-1 Benefits

  • antimicrobial
  • anti-biofilm
  • membrane-active

Tesofensine Dosing

Clinical doses: 0.25-1.0 mg orally once daily. Research typically uses 0.5 mg. Extremely long half-life (8-13 days) means steady-state in 7-10 days.

Arenicin-1 Dosing

bacterial infection|biofilm disruption

Tesofensine Side Effects

  • Dry mouth, insomnia, constipation, increased heart rate, elevated blood pressure. Not recommended with uncontrolled hypertension.

Arenicin-1 Side Effects

  • Arenicola marina

Research Overview

Tesofensine

Phase II trials showed 12.8 kg average weight loss at 1.0 mg dose over 6 months. Simultaneously inhibits reuptake of norepinephrine, dopamine, and serotonin, producing appetite suppression and increased thermogenesis.

Arenicin-1

Marine annelid peptide with strong preclinical antibacterial activity and a stable structural motif that is useful for peptide engineering.

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Common Stacking Partners

Tesofensine stacks with:

5-Amino-1MQAOD-9604MOTS-c

Arenicin-1 stacks with:

Arenicola marinabeta-hairpinantibiotic
weight-lossappetite-suppressanttriple-reuptake-inhibitorthermogenesismarine-derivedbioactiveantimicrobial peptidebiofilm