Rapamycin vs Metformin

Head-to-head comparison of Rapamycin (Rapamycin (Sirolimus)) and Metformin (Metformin Hydrochloride) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyRapamycinMetformin
CategoryAnti-AgingAnti-Aging
Full NameRapamycin (Sirolimus)Metformin Hydrochloride
Molecular Weight914.17 Da165.63 Da
Half-Life~62 hours4-8.7 hours
Amino AcidsN/AN/A
Typical Dose0.5-6 mg/week500-2000 mg/day
RouteOralOral
Purity≥98%≥98%
Studies Count15004000
Research StatusClinicalClinical

Rapamycin Benefits

  • mTOR inhibition
  • autophagy activation
  • cellular senescence modulation
  • lifespan extension in model organisms

Metformin Benefits

  • AMPK activation
  • improved insulin sensitivity
  • reduced oxidative stress
  • population-level longevity signal

Rapamycin Dosing

0.5-6 mg oral weekly in studies|intermittent dosing protocols|clinical monitoring for tolerability

Metformin Dosing

500-2000 mg/day oral|start low and titrate in trials|taken with meals

Rapamycin Side Effects

  • mouth ulcers
  • elevated lipids
  • immunosuppression
  • glucose intolerance

Metformin Side Effects

  • gastrointestinal upset
  • vitamin B12 reduction
  • diarrhea
  • rare lactic acidosis

Research Overview

Rapamycin

Rapamycin extends lifespan in multiple model organisms and is a cornerstone compound in longevity biology. Human studies focus on immune function, inflammation, and age-related biomarkers rather than proven lifespan extension.

Metformin

Metformin has extensive human data and remains a leading candidate in geroscience research. Observational and mechanistic studies suggest it may influence pathways tied to aging, though definitive anti-longevity proof in healthy humans is still lacking.

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Common Stacking Partners

Rapamycin stacks with:

MetforminSpermidineNMN

Metformin stacks with:

RapamycinNMNSpermidine
mTORautophagygerosciencelongevityAMPKinsulin-sensitivitymetabolism