MK-677 vs Macimorelin

Head-to-head comparison of MK-677 (Ibutamoren Mesylate (MK-677)) and Macimorelin (Macimorelin acetate (AEZS-130)) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyMK-677Macimorelin
CategoryGrowth HormoneGrowth Hormone
Full NameIbutamoren Mesylate (MK-677)Macimorelin acetate (AEZS-130)
Molecular Weight528.662 g/molN/A
Half-Life~24 hoursabout 4-6 hours
Amino AcidsNon-peptide compoundN/A
Typical Dose0.5 mg/kg single oral dose
RouteOral
Purity>99%≥98%
Studies Count120120
Research StatusActive ResearchClinical

MK-677 Benefits

  • Oral GH secretagogue, 24-hour GH elevation, increases IGF-1, improves sleep quality, increases lean mass, does not suppress natural GH

Macimorelin Benefits

  • diagnostic GH stimulation
  • single oral dose
  • rapid measurable GH response
  • high clinical utility

MK-677 Dosing

10-25 mg orally once daily before bedtime. 25 mg is the most studied dose. Can be used long-term without cycling.

Macimorelin Dosing

0.5 mg/kg orally as a single dose|fasted testing conditions|serial GH sampling after administration

MK-677 Side Effects

  • Increased appetite, mild water retention, drowsiness, transient numbness, mild increase in fasting blood glucose with long-term use.

Macimorelin Side Effects

  • dysgeusia or taste disturbance
  • nausea
  • headache

Research Overview

MK-677

A landmark 2-year study in elderly adults demonstrated significant increases in lean mass, GH pulsatility, and IGF-1 to youthful ranges. Selectively agonizes GHS-R1a without increasing cortisol or prolactin.

Macimorelin

Macimorelin has been validated in clinical testing as an oral alternative to injectable GH stimulation tests. Its short-term use makes it a useful translational tool for evaluating pituitary GH reserve.

Ready to buy?

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Common Stacking Partners

MK-677 stacks with:

CJC-1295IpamorelinRAD-140

Macimorelin stacks with:

Pituitary testingEndocrine workup
growth-hormone-secretagogueoralghrelin-mimeticIGF-1muscle-growthsleepdiagnosticgh-stimulation-test