Macimorelin
Macimorelin acetate (AEZS-130)
N/A Amino Acids · MW: N/A
Amino Acids
N/A
Molecular Weight
N/A
Half-life
about 4-6 hours
Research Score
4.6
Studies
120
Storage
Store lyophilized at -20°C, reconstituted at 2-8°C
What is Macimorelin?
Macimorelin is an orally active ghrelin mimetic used as a growth hormone stimulation agent. It produces a rapid GH rise after a single dose and is used clinically to help diagnose adult GH deficiency.
Key Benefits & Mechanisms
diagnostic GH stimulation
single oral dose
rapid measurable GH response
high clinical utility
Research Summary
Macimorelin has been validated in clinical testing as an oral alternative to injectable GH stimulation tests. Its short-term use makes it a useful translational tool for evaluating pituitary GH reserve.
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