Macimorelin vs Modified GRF(1-29)

Head-to-head comparison of Macimorelin (Macimorelin acetate (AEZS-130)) and Modified GRF(1-29) ([D-Ala2, Nle27]-human growth hormone-releasing hormone (1-29) amide) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyMacimorelinModified GRF(1-29)
CategoryGrowth HormoneGrowth Hormone
Full NameMacimorelin acetate (AEZS-130)[D-Ala2, Nle27]-human growth hormone-releasing hormone (1-29) amide
Molecular WeightN/AN/A
Half-Lifeabout 4-6 hours10-30 minutes
Amino AcidsN/A29
Typical Dose0.5 mg/kg single oral dose50-300 mcg
RouteOralSubcutaneous
Purity≥98%≥98%
Studies Count120150
Research StatusClinicalInvestigational

Macimorelin Benefits

  • diagnostic GH stimulation
  • single oral dose
  • rapid measurable GH response
  • high clinical utility

Modified GRF(1-29) Benefits

  • enhanced GH release
  • greater peptide stability
  • IGF-1 support research
  • longer receptor engagement

Macimorelin Dosing

0.5 mg/kg orally as a single dose|fasted testing conditions|serial GH sampling after administration

Modified GRF(1-29) Dosing

50-100 mcg SC for acute GH-response studies|100-300 mcg SC in monitored research protocols|repeat dosing in short investigative cycles with GH/IGF-1 tracking

Macimorelin Side Effects

  • dysgeusia or taste disturbance
  • nausea
  • headache

Modified GRF(1-29) Side Effects

  • headache
  • water retention
  • injection-site irritation

Research Overview

Macimorelin

Macimorelin has been validated in clinical testing as an oral alternative to injectable GH stimulation tests. Its short-term use makes it a useful translational tool for evaluating pituitary GH reserve.

Modified GRF(1-29)

Modified GRF(1-29) has been studied as a practical GHRH analog for boosting GH release while improving peptide stability versus the native fragment. It is a standard reference compound in experimental work on growth hormone pulsatility and analog design.

Ready to buy?

Find both peptides from our verified, lab-tested vendors with purity certificates and third-party testing.

Common Stacking Partners

Macimorelin stacks with:

Pituitary testingEndocrine workup

Modified GRF(1-29) stacks with:

L-arginineL-ornithineglycine
diagnosticghrelin-mimeticgh-stimulation-testghrh-analogsynthetic-peptidegrowth-hormoneresearch-compound