Macimorelin vs Capromorelin

Head-to-head comparison of Macimorelin (Macimorelin acetate (AEZS-130)) and Capromorelin (Capromorelin hydrochloride) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyMacimorelinCapromorelin
CategoryGrowth HormoneGrowth Hormone
Full NameMacimorelin acetate (AEZS-130)Capromorelin hydrochloride
Molecular WeightN/AN/A
Half-Lifeabout 4-6 hoursabout 2-3 hours
Amino AcidsN/AN/A
Typical Dose0.5 mg/kg single oral dose0.25-2 mg/kg/day
RouteOralOral
Purity≥98%≥98%
Studies Count12055
Research StatusClinicalClinical

Macimorelin Benefits

  • diagnostic GH stimulation
  • single oral dose
  • rapid measurable GH response
  • high clinical utility

Capromorelin Benefits

  • GH secretagogue activity
  • appetite stimulation
  • oral administration
  • translational animal model utility

Macimorelin Dosing

0.5 mg/kg orally as a single dose|fasted testing conditions|serial GH sampling after administration

Capromorelin Dosing

0.25-2 mg/kg orally in studies|once-daily or protocol-specific dosing|monitor appetite and body weight

Macimorelin Side Effects

  • dysgeusia or taste disturbance
  • nausea
  • headache

Capromorelin Side Effects

  • increased appetite
  • vomiting or nausea
  • lethargy

Research Overview

Macimorelin

Macimorelin has been validated in clinical testing as an oral alternative to injectable GH stimulation tests. Its short-term use makes it a useful translational tool for evaluating pituitary GH reserve.

Capromorelin

Research consistently shows capromorelin activates the ghrelin receptor pathway and increases food intake. Human development has been less prominent than veterinary use, but the compound remains a relevant GH secretagogue prototype.

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Common Stacking Partners

Macimorelin stacks with:

Pituitary testingEndocrine workup

Capromorelin stacks with:

Nutritional supportResistance training
diagnosticghrelin-mimeticgh-stimulation-testghrelin-receptor-agonistappetite-stimulantgh-secretagogue