Histatin-5 vs Elamipretide

Head-to-head comparison of Histatin-5 (Human histatin 5) and Elamipretide (Elamipretide (MTP-131, SS-31)) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyHistatin-5Elamipretide
CategoryDental & OralMuscle & Performance
Full NameHuman histatin 5Elamipretide (MTP-131, SS-31)
Molecular Weight3035 Da639.8 Da
Half-Lifeminutes in saliva1-4 hours
Amino Acids244
Typical Dose1-100 µM in research formulations0.01-0.25 mg/kg/day
RouteTopical/Oral rinseSubcutaneous/Intravenous
Purity≥98%≥98%
Studies Count120120
Research StatusPre-clinicalClinical

Histatin-5 Benefits

  • anti-Candida activity
  • biofilm suppression
  • mucosal wound support
  • oral innate immunity

Elamipretide Benefits

  • mitochondrial protection
  • reduced oxidative stress
  • improved fatigue resistance
  • may support exercise tolerance

Histatin-5 Dosing

topical rinse or gel|short contact exposure|repeat applications in research protocols

Elamipretide Dosing

0.01-0.25 mg/kg/day SC (clinical research)|daily dosing in trials|alternative IV protocols in some studies

Histatin-5 Side Effects

  • local irritation
  • proteolytic instability
  • dose-dependent cytotoxicity in vitro

Elamipretide Side Effects

  • nausea
  • injection-site reactions
  • diarrhea
  • headache

Research Overview

Histatin-5

Histatin-5 is a major salivary defense peptide that can kill Candida species and influence oral microbial communities. It is also investigated for wound-healing and xerostomia-associated oral infection models.

Elamipretide

Clinical and translational studies show elamipretide can improve mitochondrial function and some functional endpoints in mitochondrial disorders. Skeletal muscle research suggests benefits are driven by energy metabolism rather than direct muscle-building effects.

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Common Stacking Partners

Histatin-5 stacks with:

chlorhexidinefluoridexylitol

Elamipretide stacks with:

creatinecoenzyme-q10protein
antimicrobial-peptidecandidasalivaoral-defensemitochondriafatigueenergy-metabolismperformance