Histatin-5 vs ACE-031

Head-to-head comparison of Histatin-5 (Human histatin 5) and ACE-031 (ACE-031 (soluble activin receptor type IIB-Fc)) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyHistatin-5ACE-031
CategoryDental & OralMuscle & Performance
Full NameHuman histatin 5ACE-031 (soluble activin receptor type IIB-Fc)
Molecular Weight3035 Da~95 kDa
Half-Lifeminutes in salivaDays to weeks
Amino Acids24N/A
Typical Dose1-100 µM in research formulations0.1-3 mg/kg in early studies
RouteTopical/Oral rinseSubcutaneous
Purity≥98%≥98%
Studies Count12075
Research StatusPre-clinicalClinical

Histatin-5 Benefits

  • anti-Candida activity
  • biofilm suppression
  • mucosal wound support
  • oral innate immunity

ACE-031 Benefits

  • myostatin/activin neutralization
  • lean mass gain
  • muscle function support
  • anti-catabolic effect

Histatin-5 Dosing

topical rinse or gel|short contact exposure|repeat applications in research protocols

ACE-031 Dosing

Clinical studies used single or repeated SC doses|dose escalation in mg/kg|monitoring for edema/bleeding

Histatin-5 Side Effects

  • local irritation
  • proteolytic instability
  • dose-dependent cytotoxicity in vitro

ACE-031 Side Effects

  • telangiectasia/vascular effects
  • epistaxis
  • headache/edema

Research Overview

Histatin-5

Histatin-5 is a major salivary defense peptide that can kill Candida species and influence oral microbial communities. It is also investigated for wound-healing and xerostomia-associated oral infection models.

ACE-031

ACE-031 produced increases in lean mass in early studies, but development was curtailed after safety concerns and variable efficacy. Its literature remains important because it validated activin receptor blockade as a muscle-building strategy.

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Common Stacking Partners

Histatin-5 stacks with:

chlorhexidinefluoridexylitol

ACE-031 stacks with:

CreatineVitamin DLeucine
antimicrobial-peptidecandidasalivaoral-defenseactr2b-decoymyostatin-inhibitorlean-massfusion-protein