ACE-031 vs Meldonium

Head-to-head comparison of ACE-031 (ACE-031 (soluble activin receptor type IIB-Fc)) and Meldonium (3-(2,2,2-Trimethylhydrazinium)propionate) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyACE-031Meldonium
CategoryMuscle & PerformanceMuscle & Performance
Full NameACE-031 (soluble activin receptor type IIB-Fc)3-(2,2,2-Trimethylhydrazinium)propionate
Molecular Weight~95 kDa146.19 Da
Half-LifeDays to weeks~3-6 h
Amino AcidsN/AN/A
Typical Dose0.1-3 mg/kg in early studies500-1000 mg/day in divided oral doses
RouteSubcutaneousOral/IV
Purity≥98%≥98%
Studies Count7570
Research StatusClinicalClinical

ACE-031 Benefits

  • myostatin/activin neutralization
  • lean mass gain
  • muscle function support
  • anti-catabolic effect

Meldonium Benefits

  • improves exercise tolerance
  • may reduce ischemic fatigue
  • supports metabolic efficiency
  • may aid recovery

ACE-031 Dosing

Clinical studies used single or repeated SC doses|dose escalation in mg/kg|monitoring for edema/bleeding

Meldonium Dosing

500 mg orally daily|500 mg orally twice daily|500-1000 mg/day in divided doses

ACE-031 Side Effects

  • telangiectasia/vascular effects
  • epistaxis
  • headache/edema

Meldonium Side Effects

  • GI upset
  • headache
  • palpitations

Research Overview

ACE-031

ACE-031 produced increases in lean mass in early studies, but development was curtailed after safety concerns and variable efficacy. Its literature remains important because it validated activin receptor blockade as a muscle-building strategy.

Meldonium

Clinical literature focuses on cardiometabolic support and exercise tolerance rather than direct anabolic effects. Any endurance benefit is thought to come from altered substrate handling and improved tolerance to stress.

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Common Stacking Partners

ACE-031 stacks with:

CreatineVitamin DLeucine

Meldonium stacks with:

CoQ10Creatine
actr2b-decoymyostatin-inhibitorlean-massfusion-proteinmetabolic-modulatorenduranceexercise-tolerancevo2-max