Elamipretide vs Roxadustat

Head-to-head comparison of Elamipretide (Elamipretide (MTP-131, SS-31)) and Roxadustat (Roxadustat (FG-4592), hypoxia-inducible factor prolyl hydroxylase inhibitor) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyElamipretideRoxadustat
CategoryMuscle & PerformanceMuscle & Performance
Full NameElamipretide (MTP-131, SS-31)Roxadustat (FG-4592), hypoxia-inducible factor prolyl hydroxylase inhibitor
Molecular Weight639.8 Da352.35 Da
Half-Life1-4 hours~12-16 h
Amino Acids4N/A
Typical Dose0.01-0.25 mg/kg/day70-100 mg orally three times weekly
RouteSubcutaneous/IntravenousOral
Purity≥98%≥98%
Studies Count120180
Research StatusClinicalClinical

Elamipretide Benefits

  • mitochondrial protection
  • reduced oxidative stress
  • improved fatigue resistance
  • may support exercise tolerance

Roxadustat Benefits

  • induces endogenous EPO
  • improves iron handling
  • raises hemoglobin
  • may improve exercise tolerance

Elamipretide Dosing

0.01-0.25 mg/kg/day SC (clinical research)|daily dosing in trials|alternative IV protocols in some studies

Roxadustat Dosing

70-100 mg orally 3x weekly|Titrate by hemoglobin response|Monitor iron indices regularly

Elamipretide Side Effects

  • nausea
  • injection-site reactions
  • diarrhea
  • headache

Roxadustat Side Effects

  • nausea
  • hypertension
  • thrombotic events

Research Overview

Elamipretide

Clinical and translational studies show elamipretide can improve mitochondrial function and some functional endpoints in mitochondrial disorders. Skeletal muscle research suggests benefits are driven by energy metabolism rather than direct muscle-building effects.

Roxadustat

Large clinical studies support roxadustat for anemia, especially in chronic kidney disease populations. Direct VO2 max enhancement data in healthy athletes are limited, so its performance effects remain mostly inferential.

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Common Stacking Partners

Elamipretide stacks with:

creatinecoenzyme-q10protein

Roxadustat stacks with:

IronFolate
mitochondriafatigueenergy-metabolismperformancehif-stabilizererythropoiesisvo2-maxoral