Endomorphin-1 vs Insulin Glargine

Head-to-head comparison of Endomorphin-1 (Tyr-Pro-Trp-Phe-NH2) and Insulin Glargine (Insulin glargine (A21Gly,B31Arg,B32Arg human insulin analog)) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyEndomorphin-1Insulin Glargine
CategoryPain ManagementDiabetes & Metabolic
Full NameTyr-Pro-Trp-Phe-NH2Insulin glargine (A21Gly,B31Arg,B32Arg human insulin analog)
Molecular Weight610.71 Da6063.6 Da
Half-LifeMinutes in plasmaAbout 12-24 hours
Amino Acids451
Typical Dose0.1-10 ug per animal0.1-0.2 U/kg once daily
RouteIntrathecal / subcutaneousSubcutaneous
Purity≥98%≥98%
Studies Count60013000
Research StatusPre-clinicalApproved

Endomorphin-1 Benefits

  • mu-opioid selectivity
  • potent antinociception
  • endogenous peptide scaffold
  • useful for receptor-discovery studies

Insulin Glargine Benefits

  • Once-daily basal coverage
  • Smooth action profile
  • Lower nocturnal hypoglycemia risk
  • Improves fasting glucose control

Endomorphin-1 Dosing

Intrathecal 0.1-10 ug per animal|Subcutaneous 0.1-5 ug per animal|In vitro 0.1-100 nM

Insulin Glargine Dosing

Inject SC once daily at the same time each day|Titrate every 3-4 days to fasting glucose targets|Can be combined with prandial insulin

Endomorphin-1 Side Effects

  • respiratory depression at high exposure
  • sedation
  • tolerance and dependence potential

Insulin Glargine Side Effects

  • Hypoglycemia
  • Injection-site reactions
  • Weight gain

Research Overview

Endomorphin-1

Endomorphin-1 is a key research peptide in studies of endogenous mu-opioid signaling and spinal analgesia. Like other peptide analgesics, its main translational hurdles are enzymatic instability, limited oral bioavailability, and delivery across barriers.

Insulin Glargine

Clinical and translational studies support its use as a basal comparator because of prolonged absorption and stable glycemic control. It is heavily used in basal-bolus regimen research and insulin-delivery optimization studies.

Ready to buy?

Find both peptides from our verified, lab-tested vendors with purity certificates and third-party testing.

Common Stacking Partners

Endomorphin-1 stacks with:

gabapentinketamine

Insulin Glargine stacks with:

Insulin LisproInsulin Aspart
mu-opioidendogenous-peptideanalgesiapain-modulationbasal insulinlong-actingfasting glucose