DPDPE vs Cosyntropin

Head-to-head comparison of DPDPE ([D-Pen2, D-Pen5]-enkephalin) and Cosyntropin (Cosyntropin (ACTH 1-24)) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyDPDPECosyntropin
CategoryPain ManagementPain Management
Full Name[D-Pen2, D-Pen5]-enkephalinCosyntropin (ACTH 1-24)
Molecular Weight645.79 Da2933.3 Da
Half-Life15-60 minutes in plasma~10 min
Amino Acids524
Typical Dose0.01-1 ug per animal0.25 mg IV/IM diagnostic dose|off-label headache protocols vary
RouteIntrathecal / intracerebroventricularIV|IM
Purity≥98%≥98%
Studies Count80061
Research StatusPre-clinicalClinical research

DPDPE Benefits

  • delta-opioid selectivity
  • improved conformational stability
  • analgesic receptor mapping
  • useful in chronic pain models

Cosyntropin Benefits

  • refractory migraine
  • anti-inflammatory signaling
  • headache rescue research

DPDPE Dosing

Intrathecal 0.01-1 ug per animal|Intracerebroventricular 0.01-0.5 ug per animal|In vitro 0.1-20 nM

Cosyntropin Dosing

0.25 mg IV/IM|1 mg IV/IM

DPDPE Side Effects

  • sedation
  • nausea-like opioid effects
  • tolerance with repeated dosing

Cosyntropin Side Effects

  • flushing
  • nausea

Research Overview

DPDPE

DPDPE is widely cited in opioid pharmacology because it helped establish the functional role of delta-opioid receptors in pain control. Its constrained structure is also used to explore how peptide cyclization changes potency, stability, and tissue selectivity.

Cosyntropin

Cosyntropin is not a standard pain drug, but it appears in headache literature because ACTH analogs can help some patients with difficult migraine attacks. The analgesic rationale is partly tied to steroidogenic and anti-inflammatory effects.

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Common Stacking Partners

DPDPE stacks with:

morphinegabapentin

Cosyntropin stacks with:

ACTH(1-24)Synacthen
cyclic-peptidedelta-opioidanalgesiaenkephalin-analogmigraineheadacheACTH-analog