Cholecystokinin-8 vs Macimorelin

Head-to-head comparison of Cholecystokinin-8 (Cholecystokinin (sulfated C-terminal octapeptide, CCK-8)) and Macimorelin (Macimorelin acetate (AEZS-130)) — benefits, dosing, side effects, research data, and where to buy.

PropertyCholecystokinin-8Macimorelin
CategoryEndocrine PeptidesGrowth Hormone
Full NameCholecystokinin (sulfated C-terminal octapeptide, CCK-8)Macimorelin acetate (AEZS-130)
Molecular Weight1143.2 DaN/A
Half-Life1-2 minabout 4-6 hours
Amino AcidsDY(SO3H)MGWMDF-NH2N/A
Typical Dosephysiologic low-picomolar-nanomolar range|research-dependent0.5 mg/kg single oral dose
Routeendogenous secretion|research IV/SCOral
Purity≥98%≥98%
Studies Count97120
Research StatusEndogenousClinical

Cholecystokinin-8 Benefits

  • gallbladder contraction
  • pancreatic enzyme release
  • satiety signaling

Macimorelin Benefits

  • diagnostic GH stimulation
  • single oral dose
  • rapid measurable GH response
  • high clinical utility

Cholecystokinin-8 Dosing

physiologic secretion|research-dependent

Macimorelin Dosing

0.5 mg/kg orally as a single dose|fasted testing conditions|serial GH sampling after administration

Cholecystokinin-8 Side Effects

  • abdominal cramping
  • nausea
  • biliary contraction

Macimorelin Side Effects

  • dysgeusia or taste disturbance
  • nausea
  • headache

Research Overview

Cholecystokinin-8

CCK-8 is a canonical gut hormone fragment with extensive documentation in digestive physiology and appetite control. Sulfation of the tyrosine residue is important for high-affinity receptor activity.

Macimorelin

Macimorelin has been validated in clinical testing as an oral alternative to injectable GH stimulation tests. Its short-term use makes it a useful translational tool for evaluating pituitary GH reserve.

Ready to buy?

Find both peptides from our verified, lab-tested vendors with purity certificates and third-party testing.

Common Stacking Partners

Cholecystokinin-8 stacks with:

gallbladderpancreassatiety

Macimorelin stacks with:

Pituitary testingEndocrine workup
gut-hormonesatiety-peptideendocrine-peptidediagnosticghrelin-mimeticgh-stimulation-test