Cholecystokinin-8 vs Bremelanotide

Head-to-head comparison of Cholecystokinin-8 (Cholecystokinin (sulfated C-terminal octapeptide, CCK-8)) and Bremelanotide (Bremelanotide (PT-141), cyclic melanocortin receptor agonist) — benefits, dosing, side effects, research data, and where to buy.

PropertyCholecystokinin-8Bremelanotide
CategoryEndocrine PeptidesSexual Health
Full NameCholecystokinin (sulfated C-terminal octapeptide, CCK-8)Bremelanotide (PT-141), cyclic melanocortin receptor agonist
Molecular Weight1143.2 Da1025.2 Da
Half-Life1-2 minabout 2.7 h
Amino AcidsDY(SO3H)MGWMDF-NH27
Typical Dosephysiologic low-picomolar-nanomolar range|research-dependent1.75 mg
Routeendogenous secretion|research IV/SCSubcutaneous
Purity≥98%≥98%
Studies Count97200
Research StatusEndogenousClinical

Cholecystokinin-8 Benefits

  • gallbladder contraction
  • pancreatic enzyme release
  • satiety signaling

Bremelanotide Benefits

  • increases sexual desire
  • supports arousal
  • may improve erectile response
  • on-demand use

Cholecystokinin-8 Dosing

physiologic secretion|research-dependent

Bremelanotide Dosing

1.75 mg subcutaneous PRN|administer about 45 minutes before activity|max 1 dose per 24 hours

Cholecystokinin-8 Side Effects

  • abdominal cramping
  • nausea
  • biliary contraction

Bremelanotide Side Effects

  • nausea
  • flushing
  • headache
  • transient blood pressure increase

Research Overview

Cholecystokinin-8

CCK-8 is a canonical gut hormone fragment with extensive documentation in digestive physiology and appetite control. Sulfation of the tyrosine residue is important for high-affinity receptor activity.

Bremelanotide

Human studies and approval data support meaningful effects on sexual desire in women, with a central mechanism involving melanocortin signaling. It is one of the most clinically relevant peptides in this category and is commonly used as the reference compound for PT-141-type research.

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Common Stacking Partners

Cholecystokinin-8 stacks with:

gallbladderpancreassatiety

Bremelanotide stacks with:

Kisspeptin-54Melanotan-II
gut-hormonesatiety-peptideendocrine-peptidemelanocortinlibidoerectile-functionapproved