C-peptide vs Macimorelin

Head-to-head comparison of C-peptide (Connecting peptide (C-peptide)) and Macimorelin (Macimorelin acetate (AEZS-130)) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyC-peptideMacimorelin
CategoryPain ManagementGrowth Hormone
Full NameConnecting peptide (C-peptide)Macimorelin acetate (AEZS-130)
Molecular Weight3020.3 DaN/A
Half-Life~20-30 minabout 4-6 hours
Amino Acids31N/A
Typical Doseno approved analgesic dose|research-only0.5 mg/kg single oral dose
RouteIV|subQOral
Purity≥98%≥98%
Studies Count46120
Research StatusPre-clinicalClinical

C-peptide Benefits

  • diabetic neuropathy research
  • nerve function support
  • possible analgesic effect

Macimorelin Benefits

  • diagnostic GH stimulation
  • single oral dose
  • rapid measurable GH response
  • high clinical utility

C-peptide Dosing

0.5-1.0 mg/day in research|route varies by protocol

Macimorelin Dosing

0.5 mg/kg orally as a single dose|fasted testing conditions|serial GH sampling after administration

C-peptide Side Effects

  • injection-site reactions
  • unknown long-term safety

Macimorelin Side Effects

  • dysgeusia or taste disturbance
  • nausea
  • headache

Research Overview

C-peptide

C-peptide is not an approved analgesic, but multiple studies have examined its effects on peripheral nerve blood flow and neuropathy outcomes. The strongest relevance is in diabetic neuropathic pain rather than migraine.

Macimorelin

Macimorelin has been validated in clinical testing as an oral alternative to injectable GH stimulation tests. Its short-term use makes it a useful translational tool for evaluating pituitary GH reserve.

Ready to buy?

Find both peptides from our verified, lab-tested vendors with purity certificates and third-party testing.

Common Stacking Partners

C-peptide stacks with:

C-peptideConnecting peptide

Macimorelin stacks with:

Pituitary testingEndocrine workup
neuropathic-paindiabetic-neuropathynerve-repairdiagnosticghrelin-mimeticgh-stimulation-test