Plitidepsin vs Mambalgin-1

Head-to-head comparison of Plitidepsin (Dehydrodidemnin B (Plitidepsin)) and Mambalgin-1 (Mambalgin-1 from Dendroaspis polylepis venom) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyPlitidepsinMambalgin-1
CategoryExperimentalExperimental
Full NameDehydrodidemnin B (Plitidepsin)Mambalgin-1 from Dendroaspis polylepis venom
Molecular Weight1110.3 Da6,300 Da
Half-LifeApproximately 44 hoursMinutes to hours
Amino AcidsN/A57
Typical Dose1.5 mg/m2 IV0.1-1 nmol intrathecal|10-100 nM in vitro|single-dose rodent studies
RouteIntravenousIntrathecal
Purity≥98%≥98%
Studies Count24055
Research StatusClinicalPre-clinical

Plitidepsin Benefits

  • antineoplastic
  • antiviral
  • pro-apoptotic
  • anti-inflammatory

Mambalgin-1 Benefits

  • ASIC channel inhibition
  • non-opioid analgesia research
  • sensory-neuron physiology
  • lead optimization for pain therapeutics

Plitidepsin Dosing

1.5 mg/m2 IV infusion in oncology trials|q21d or similar intermittent schedules|dose escalation and combination protocols in studies

Mambalgin-1 Dosing

Intrathecal pain-behavior studies|ASIC1a/ASIC1b electrophysiology|Acute dosing in rodents

Plitidepsin Side Effects

  • nausea
  • fatigue
  • transaminase elevation

Mambalgin-1 Side Effects

  • Hypoactivity at high dose
  • off-target ASIC blockade
  • local irritation

Research Overview

Plitidepsin

Plitidepsin has been studied for its ability to disrupt eEF1A-dependent pathways, induce oxidative stress, and suppress tumor cell growth. It has reached clinical oncology development and was also evaluated as a candidate against SARS-CoV-2 in the literature.

Mambalgin-1

Pre-clinical work shows mambalgin-1 can reduce pain behaviors by modulating proton-gated ion channels in peripheral and central pathways. It has become an important template for developing ASIC-targeted analgesics.

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Common Stacking Partners

Plitidepsin stacks with:

dexamethasonebortezomibgemcitabine

Mambalgin-1 stacks with:

gabapentinbaclofenlidocaine
marine-derivedtunicatedepsipeptideanticancersnake-venomthree-finger-toxinasic-blockerpain-research