P11-4 vs Endomorphin-1

Head-to-head comparison of P11-4 (Self-assembling peptide P11-4 (Ac-QQRFEWEFEQQ-NH2)) and Endomorphin-1 (Tyr-Pro-Trp-Phe-NH2) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyP11-4Endomorphin-1
CategoryDental & OralPain Management
Full NameSelf-assembling peptide P11-4 (Ac-QQRFEWEFEQQ-NH2)Tyr-Pro-Trp-Phe-NH2
Molecular Weight1466 Da610.71 Da
Half-Lifelocal activity for hours; peptide degraded over timeMinutes in plasma
Amino Acids114
Typical Dose0.5-5 mg per lesion0.1-10 ug per animal
RouteTopical/IntraoralIntrathecal / subcutaneous
Purity≥98%≥98%
Studies Count40600
Research StatusClinicalPre-clinical

P11-4 Benefits

  • enamel remineralization
  • early caries arrest
  • biomimetic scaffold formation
  • minimally invasive repair

Endomorphin-1 Benefits

  • mu-opioid selectivity
  • potent antinociception
  • endogenous peptide scaffold
  • useful for receptor-discovery studies

P11-4 Dosing

topical application to cleaned lesion|single-visit in-office application|repeat at follow-up if indicated

Endomorphin-1 Dosing

Intrathecal 0.1-10 ug per animal|Subcutaneous 0.1-5 ug per animal|In vitro 0.1-100 nM

P11-4 Side Effects

  • transient tooth sensitivity
  • local irritation
  • taste disturbance

Endomorphin-1 Side Effects

  • respiratory depression at high exposure
  • sedation
  • tolerance and dependence potential

Research Overview

P11-4

P11-4 has been studied for its ability to penetrate initial carious lesions and self-assemble into a fibrillar matrix that nucleates hydroxyapatite. Human and preclinical studies support its role in non-invasive enamel repair.

Endomorphin-1

Endomorphin-1 is a key research peptide in studies of endogenous mu-opioid signaling and spinal analgesia. Like other peptide analgesics, its main translational hurdles are enzymatic instability, limited oral bioavailability, and delivery across barriers.

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Common Stacking Partners

P11-4 stacks with:

fluoride varnishCPP-ACPxylitol

Endomorphin-1 stacks with:

gabapentinketamine
enamel-remineralizationcariesbiomimetic-peptideoral-healthmu-opioidendogenous-peptideanalgesiapain-modulation