Orexin-A vs Tianeptine sodium

Head-to-head comparison of Orexin-A (Hypocretin-1 (Orexin-A)) and Tianeptine sodium (Tianeptine sodium) — benefits, dosing, side effects, research data, and where to buy.

PropertyOrexin-ATianeptine sodium
CategoryCognitive EnhancementCognitive Enhancement
Full NameHypocretin-1 (Orexin-A)Tianeptine sodium
Molecular Weight3562 Da458.94 Da
Half-LifeMinutes to <1 hourAbout 2.5 hours
Amino Acids33N/A
Typical DoseResearch-only; no validated human dose12.5 mg 3 times daily
RouteIntracerebroventricular/IntranasalOral
Purity≥98%≥98%
Studies Count42280
Research StatusPre-clinicalClinical

Orexin-A Benefits

  • wakefulness
  • attention
  • memory consolidation
  • fatigue resistance

Tianeptine sodium Benefits

  • mood improvement
  • anxiety reduction
  • cognitive clarity
  • stress adaptation

Orexin-A Dosing

Research-only i.c.v. microgram/nanomolar studies|intranasal experimental use|no established human protocol

Tianeptine sodium Dosing

12.5 mg oral 3x/day|25 mg/day oral|clinical antidepressant dosing

Orexin-A Side Effects

  • insomnia
  • headache
  • blood pressure changes

Tianeptine sodium Side Effects

  • nausea
  • dizziness
  • dependence risk

Research Overview

Orexin-A

Preclinical studies link orexin signaling to arousal, learning, and memory consolidation, making orexin-A a candidate for cognition-related research. It is not an approved cognitive enhancer and remains an experimental peptide.

Tianeptine sodium

Clinical studies support tianeptine as an antidepressant with a distinctive glutamatergic and neuroplasticity-related profile. Some evidence suggests cognitive benefits in mood-impaired populations, likely secondary to improved stress handling and affect.

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Common Stacking Partners

Orexin-A stacks with:

PRL-8-53Bromantane

Tianeptine sodium stacks with:

BromantanePRL-8-53
peptidewakefulnessmemoryantidepressantanxiolyticmood