Tianeptine sodium vs NPY

Head-to-head comparison of Tianeptine sodium (Tianeptine sodium) and NPY (Neuropeptide Y) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyTianeptine sodiumNPY
CategoryCognitive EnhancementCognitive Enhancement
Full NameTianeptine sodiumNeuropeptide Y
Molecular Weight458.94 Da4272 Da
Half-LifeAbout 2.5 hoursminutes
Amino AcidsN/A36 aa
Typical Dose12.5 mg 3 times daily1-10 µg preclinical range
RouteOralIntranasal
Purity≥98%≥98%
Studies Count280900
Research StatusClinicalPre-clinical

Tianeptine sodium Benefits

  • mood improvement
  • anxiety reduction
  • cognitive clarity
  • stress adaptation

NPY Benefits

  • stress resilience
  • hippocampal protection
  • memory modulation
  • anti-excitotoxic signaling

Tianeptine sodium Dosing

12.5 mg oral 3x/day|25 mg/day oral|clinical antidepressant dosing

NPY Dosing

0.1-1 nmol ICV in rodents|1-10 µg intranasal in experimental work|acute or repeated stress-model protocols

Tianeptine sodium Side Effects

  • nausea
  • dizziness
  • dependence risk

NPY Side Effects

  • sedation
  • appetite increase
  • blood pressure changes

Research Overview

Tianeptine sodium

Clinical studies support tianeptine as an antidepressant with a distinctive glutamatergic and neuroplasticity-related profile. Some evidence suggests cognitive benefits in mood-impaired populations, likely secondary to improved stress handling and affect.

NPY

NPY has been shown in animal studies to protect neurons from excitotoxic injury and to dampen stress-linked cognitive impairment. It is often discussed as a counterbalance to overactive glutamatergic and stress pathways in the brain.

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Common Stacking Partners

Tianeptine sodium stacks with:

BromantanePRL-8-53

NPY stacks with:

magnesium-threonateciticolinebacopa
antidepressantanxiolyticmoodstresshippocampusneuroprotectionmemory