Met-enkephalin vs P11-4

Head-to-head comparison of Met-enkephalin (Tyr-Gly-Gly-Phe-Met) and P11-4 (Self-assembling peptide P11-4 (Ac-QQRFEWEFEQQ-NH2)) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyMet-enkephalinP11-4
CategoryPain ManagementDental & Oral
Full NameTyr-Gly-Gly-Phe-MetSelf-assembling peptide P11-4 (Ac-QQRFEWEFEQQ-NH2)
Molecular Weight573.67 Da1466 Da
Half-Life1-5 minutes in plasmalocal activity for hours; peptide degraded over time
Amino Acids511
Typical Dose0.1-5 ug per animal0.5-5 mg per lesion
RouteIntrathecal / intracerebroventricularTopical/Intraoral
Purity≥98%≥98%
Studies Count120040
Research StatusPre-clinicalClinical

Met-enkephalin Benefits

  • endogenous opioid signaling
  • analgesic reference ligand
  • spinal antinociception
  • neurochemical pain-pathway probe

P11-4 Benefits

  • enamel remineralization
  • early caries arrest
  • biomimetic scaffold formation
  • minimally invasive repair

Met-enkephalin Dosing

Intrathecal 0.1-5 ug per animal|Intracerebroventricular 0.1-2 ug per animal|In vitro 1-100 nM

P11-4 Dosing

topical application to cleaned lesion|single-visit in-office application|repeat at follow-up if indicated

Met-enkephalin Side Effects

  • sedation at higher exposure
  • constipation-like opioid effects
  • rapid enzymatic degradation

P11-4 Side Effects

  • transient tooth sensitivity
  • local irritation
  • taste disturbance

Research Overview

Met-enkephalin

Met-enkephalin has been extensively used in receptor pharmacology and nociception studies to map mu and delta opioid biology. The main limitation in translational work is very short half-life from peptidase cleavage and poor systemic stability.

P11-4

P11-4 has been studied for its ability to penetrate initial carious lesions and self-assemble into a fibrillar matrix that nucleates hydroxyapatite. Human and preclinical studies support its role in non-invasive enamel repair.

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Common Stacking Partners

Met-enkephalin stacks with:

gabapentinketamine

P11-4 stacks with:

fluoride varnishCPP-ACPxylitol
opioid-peptideenkephalinmu-opioidanalgesiaenamel-remineralizationcariesbiomimetic-peptideoral-health